SCHEMBL1551925

SCHEMBL1551925

Oc1ccc[c]c1Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 1/20 0.45
BCL2L1 Q07817 1/20 0.45
IDH1 O75874 1/20 0.42
CALM1 P0DP23 1/20 0.42
ALOX5 P09917 1/20 0.40
KEAP1 Q14145 1/20 0.38
MEN1 O00255 1/20 0.38
CYP3A4 P08684 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
KMT2A Q03164 1/20 0.38
HIF1A Q16665 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HNF4A P41235 1/20 0.37
HSPA5 P11021 1/20 0.37
CHUK O15111 1/20 0.36
TXNRD1 Q16881 1/20 0.36
NOX4 Q9NPH5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27561165 0.83 TRPA1 (0.38) IDH1ALOX5KEAP1MEN1HPGD
SCHEMBL16720697 0.82 KDM4E (0.43) KEAP1HPGDALOX15HSD17B10
SCHEMBL8802600 0.78 BCL2 (0.44) BCL2BCL2L1IDH1CALM1ALOX5
SCHEMBL8466360 0.78 CALM1 (0.55) BCL2BCL2L1IDH1CALM1CYP3A4
SCHEMBL7465411 0.78 CALM1 (0.44) BCL2BCL2L1CALM1MEN1CYP3A4
SCHEMBL721135 0.78 CALM1 (0.44) BCL2BCL2L1CALM1ALOX5KEAP1
SCHEMBL27703315 0.77 KDM4E (0.43) MEN1HPGDALOX15KMT2AHSD17B10
SCHEMBL7459473 0.76 CALM1 (0.42) BCL2BCL2L1CALM1ALOX5MEN1
SCHEMBL28815316 0.76 CALM1 (0.42) CALM1CYP3A4ALOX15
SCHEMBL7453243 0.76 CALM1 (0.42) BCL2BCL2L1IDH1CALM1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE46830-E1 Method for solid phase peptide synthesis POLYPEPTIDE LABORATORIES HOLDING (PPL) AB (SE) 2018-05-08 US disclosed
US-20170283478-A1 PROCESS FOR PREPARATION OF LIRAGLUTIDE DR. REDDY'S LABORATORIES LIMITED (IN) 2017-10-05 US disclosed
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2016005960-A1 PROCESS FOR PREPARATION OF LIRAGLUTIDE DR. REDDY'S LABORATORIES LIMITED (IN) 2016-01-14 WO disclosed
US-9040480-B2 Synthesis of glucagon-like peptide LONZA AG (CH) 2015-05-26 US disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed
US-20130324699-A1 SYNTHESIS OF GLUCAGON-LIKE PEPTIDE LONZA AG (CH) 2013-12-05 US disclosed
US-8445433-B2 Synthesis of glucagon-like peptide LONZA AG (CH) 2013-05-21 US disclosed
US-7939629-B2 Method for solid phase peptide synthesis LONZA AG (CH) 2011-05-10 US disclosed
EP-1987052-B1 SYNTHESIS OF GLUCAGON-LIKE PEPTIDES LONZA AG (CH) 2011-04-27 EP disclosed
WO-2006032457-A9 PEPTIDE CYCLISATION LONZA AG (CH) 2006-05-26 WO disclosed
WO-2006045503-A1 METHOD FOR SOLID PHASE PEPTIDE SYNTHESIS LONZA AG (CH) 2006-05-04 WO disclosed
WO-2006032457-A1 PEPTIDE CYCLISATION LONZA AG (CH) 2006-03-30 WO disclosed
EP-0848694-A4 REDUCING ESTROGENICITY OF ALKOXYLATED COMPOUNDS AND PRODUCTS THEREOF WITCO CORP (US) 1999-08-25 EP disclosed
EP-0848694-A1 REDUCING ESTROGENICITY OF ALKOXYLATED COMPOUNDS AND PRODUCTS THEREOF WITCO CORPORATION (US) 1998-06-24 EP disclosed
EP-0804191-A1 TREATMENT OF PLATELET DERIVED GROWTH FACTOR RELATED DISORDERS SUCH AS CANCERS USING INHIBITORS OF PLATELET DERIVED GROWTH RECEPTOR Sugen, Inc. (US) 1997-11-05 EP disclosed
WO-1997006125-A1 REDUCING ESTROGENICITY OF ALKOXYLATED COMPOUNDS AND PRODUCTS THEREOF WITCO CORPORATION (US) 1997-02-20 WO disclosed
WO-1995019169-A2 TREATMENT OF PLATELET DERIVED GROWTH FACTOR RELATED DISORDERS SUCH AS CANCER USING INHIBITORS OF PLATELET DERIVED GROWTH FACTOR RECEPTOR SUGEN, INC. (US) 1995-07-20 WO disclosed
US-4605759-A ACIDIFYING THE REACTION PRODUCT OF GLYCINE, A BENZALDEHYDE AND GROUP 1 METAL HYDROXIDE USING WATER/SOLVENT MIXTURE AND A PHASE TRANSFER AGENT MITSUI TOATSU CHEMICALS, INC. (JP) 1986-08-12 US disclosed
EP-0051023-A1 Derivatives of the benzoyl and alpha hydroxybenzyl-phenyl osides family, method for their preparation and their therapeutic application SOCIETE DE RECHERCHES INDUSTRIELLES S.O.R.I. Société anonyme dite: (FR) 1982-05-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130324699-A1 SYNTHESIS OF GLUCAGON-LIKE PEPTIDE GLP1R, IAPP, GIPR BCL2 4033/4885BCL2L1 2222/4885IDH1 2790/4885
US-20170283478-A1 PROCESS FOR PREPARATION OF LIRAGLUTIDE GLP1R, IAPP, GCG BCL2 2759/4885BCL2L1 2977/4885IDH1 4067/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.