SCHEMBL15519612

SCHEMBL15519612

NC(=O)N(c1ccc(O)cc1)c1ccn[nH]1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.34
ESR1 P03372 7/20 0.33
ESR2 Q92731 7/20 0.33
CA2 P00918 1/20 0.31
PEPD P12955 1/20 0.31
MPO P05164 1/20 0.31
CYP3A4 P08684 1/20 0.31
KDM5A P29375 1/20 0.31
BLM P54132 1/20 0.31
GFER P55789 1/20 0.31
PMP22 Q01453 1/20 0.31
HIF1A Q16665 1/20 0.31
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11417635 0.76 ESR1 (0.43) ESR1ESR2CA2PEPDMPO
SCHEMBL15519775 0.75 NNMT (0.44)
SCHEMBL5533968 0.71 NPSR1 (0.45) HCAR2CA2NPC1RAB9A
SCHEMBL1013105 0.71 TRPM8 (0.39) HCAR2
SCHEMBL4561593 0.70 HCAR2 (0.39) HCAR2NPC1RAB9A
SCHEMBL27584809 0.70 HCAR2 (0.33) HCAR2ESR1ESR2
SCHEMBL27296095 0.70 NPSR1 (0.52) ESR1ESR2CA2NPC1RAB9A
SCHEMBL6037486 0.68 ACHE (0.52) ESR1ESR2CA2PEPDNPC1
SCHEMBL15542608 0.68 HCAR2 (0.37) HCAR2NPC1RAB9A
SCHEMBL27537276 0.66 HCAR2 (0.38) HCAR2MPOCYP3A4NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2890693-A1 PYRAZOLE DERIVATIVES AS P38 MAP INHIBITORS Respivert Limited (GB) 2015-07-08 EP claimed
WO-2014033448-A1 PYRAZOLE DERIVATIVES AS P38 MAP INHIBITORS RESPIVERT LIMTED (GB) 2014-03-06 WO claimed