SCHEMBL15520532

SCHEMBL15520532

CC(c1ccc(-c2ccc(F)c(OC(=O)O)c2)cc1Cl)C(O)(c1ccc2c(c1)N(C)C(=O)CO2)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR55 Q9Y2T6 1/20 0.38
ALDH1A1 P00352 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
KMO O15229 3/20 0.32
BRD4 O60885 1/20 0.32
USP2 O75604 1/20 0.32
HTT P42858 1/20 0.32
TSHR P16473 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
THRB P10828 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
SLC5A1 P13866 1/20 0.30
SLC5A2 P31639 1/20 0.30
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30
CTSC P53634 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15520752 0.95 GPR55 (0.38) GPR55ALDH1A1PDE3BPDE3AKMO
SCHEMBL15520803 0.95 GPR55 (0.38) GPR55ALDH1A1PDE3BPDE3AKMO
SCHEMBL15520533 0.95 GPR55 (0.38) GPR55ALDH1A1PDE3BPDE3AKMO
SCHEMBL15520206 0.94 GPR55 (0.37) GPR55ALDH1A1PDE3BPDE3AKMO
SCHEMBL15520371 0.93 GPR55 (0.37) GPR55ALDH1A1PDE3BPDE3AKMO
SCHEMBL15520843 0.92 GPR55 (0.36) GPR55ALDH1A1PDE3BPDE3AKMO
SCHEMBL15520261 0.91 USP2 (0.40) ALDH1A1KMOBRD4USP2HTT
SCHEMBL15519642 0.90 GPR55 (0.37) GPR55ALDH1A1PDE3BPDE3AKMO
SCHEMBL15520365 0.89 FFAR4 (0.35) GPR55ALDH1A1PDE3BPDE3AKMO
SCHEMBL15520262 0.89 GPR55 (0.36) GPR55ALDH1A1PDE3BPDE3AKMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP claimed