SCHEMBL15526366

SCHEMBL15526366

CCCCCCCCCCCCCCCC(=O)OCC(COC(=O)CCCCCCCCCCCCCCC)OP(=O)(O)OCCN

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 8/20 0.59
LPAR3 Q9UBY5 7/20 0.57
LPAR1 Q92633 6/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
PLA2G2C Q5R387 1/20 0.57
FABP3 P05413 1/20 0.57
LPAR6 P43657 3/20 0.54
LPAR4 Q99677 3/20 0.54
LPAR5 Q9H1C0 3/20 0.54
LPAR2 Q9HBW0 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1402383 1.00 ENPP2 (0.59) ENPP2LPAR3LPAR1SMN1; SMN2PLA2G2C
SCHEMBL6254776 0.94 PRKCA (0.56) ENPP2LPAR3LPAR1SMN1; SMN2FABP3
SCHEMBL7204294 0.94 PRKCA (0.56) ENPP2LPAR3LPAR1SMN1; SMN2FABP3
SCHEMBL14659956 0.94 PRKCA (0.56) ENPP2LPAR3LPAR1SMN1; SMN2FABP3
SCHEMBL19629017 0.94 ENPP2 (0.57) ENPP2LPAR3LPAR1SMN1; SMN2FABP3
SCHEMBL16714278 0.93 ENPP2 (0.64) ENPP2LPAR3LPAR1
SCHEMBL190727 0.93 ENPP2 (0.64) ENPP2LPAR3LPAR1
SCHEMBL18719361 0.91 ENPP2 (0.63) ENPP2LPAR3LPAR1SMN1; SMN2FABP3
SCHEMBL2126025 0.88 PRKCE (0.61) ENPP2LPAR3
SCHEMBL3645476 0.87 ENPP2 (0.57) ENPP2LPAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 75 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4667492-A2 TARGETED LIPID PARTICLES FOR SYSTEMIC DELIVERY OF NUCLEIC ACID MOLECULES TO LEUKOCYTES Ramot at Tel-Aviv University Ltd. (IL) 2025-12-24 EP claimed
WO-2025242657-A1 LIPOPEPTIDE BUILDING BLOCKS AND AGGREGATES SHAPE BIOPHARMACEUTICALS AG (CH) 2025-11-27 WO claimed
EP-4615416-A1 SELF-ASSEMBLING LIPID NANOPARTICLES FOR TARGETED DELIVERY OF THERAPEUTIC AGENTS Ramot at Tel-Aviv University Ltd. (IL) 2025-09-17 EP claimed
EP-3160448-B1 LIPOSOMAL FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS UNIV RAMOT (IL) 2025-08-06 EP claimed
EP-3303598-B1 TARGETED LIPID PARTICLES FOR SYSTEMIC DELIVERY OF NUCLEIC ACID MOLECULES TO LEUKOCYTES UNIV RAMOT (IL) 2025-03-19 EP claimed
WO-2025049765-A1 TARGETING LIPID NANOPARTICLES FOR NUCLEIC ACID DELIVERY EMD MILLIPORE CORPORATION (US) 2025-03-06 WO claimed
WO-2025029640-A1 TARGETING LIPOSOME FOR PROTEIN DEGRADER DELIVERY SIGMA-ALDRICH CO. LLC (US) 2025-02-06 WO claimed
US-12065664-B2 Method for treatment of a leukocyte related disease by delivery of nucleic acid molecules to leukocytes using targeted lipid particles RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2024-08-20 US claimed
WO-2024100656-A1 SELF-ASSEMBLING LIPID NANOPARTICLES FOR TARGETED DELIVERY OF THERAPEUTIC AGENTS RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2024-05-16 WO claimed
WO-2022103927-A1 IMMUNOGENIC COMPOSITIONS FOR CORONAVIRUSES SHAPE BIOPHARMACEUTICALS INC. (US) 2022-05-19 WO claimed
US-20210108228-A1 TARGETED LIPID PARTICLES FOR SYSTEMIC DELIVERY OF NUCLEIC ACID MOLECULES TO LEUKOCYTES RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2021-04-15 US claimed
EP-2839015-B1 LIPIDATED GLYCOSAMINOGLYCAN PARTICLES FOR THE DELIVERY OF NUCLEIC ACIDS UNIV RAMOT (IL) 2020-04-29 EP claimed
US-10583084-B2 Liposomal formulations for delivery of nucleic acids RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2020-03-10 US claimed
US-20180142261-A1 TARGETED LIPID PARTICLES FOR SYSTEMIC DELIVERY OF NUCLEIC ACID MOLECULES TO LEUKOCYTES RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2018-05-24 US claimed
EP-3303598-A1 TARGETED LIPID PARTICLES FOR SYSTEMIC DELIVERY OF NUCLEIC ACID MOLECULES TO LEUKOCYTES Ramot at Tel-Aviv University Ltd. (IL) 2018-04-11 EP claimed
US-20170128367-A1 LIPOSOMAL FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2017-05-11 US claimed
EP-3160448-A1 LIPOSOMAL FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS Ramot at Tel-Aviv University Ltd. (IL) 2017-05-03 EP claimed
WO-2016189532-A1 TARGETED LIPID PARTICLES FOR SYSTEMIC DELIVERY OF NUCLEIC ACID MOLECULES TO LEUKOCYTES RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2016-12-01 WO claimed
WO-2015198326-A1 LIPOSOMAL FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2015-12-30 WO claimed
US-20150140108-A1 LIPIDATED GLYCOSAMINOGLYCAN PARTICLES FOR THE DELIVERY OF NUCLEIC ACIDS RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2015-05-21 US claimed