SCHEMBL15531012

SCHEMBL15531012

O=C(Nc1ccnnc1)C1CNC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KHK P50053 2/20 0.40
RORC P51449 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.39
ABL1 P00519 1/20 0.39
ROCK2 O75116 3/20 0.39
ROCK1 Q13464 3/20 0.39
PARP1 P09874 3/20 0.39
DYRK1A Q13627 3/20 0.38
RPS6KA5 O75582 2/20 0.38
PKN2 Q16513 2/20 0.38
LRRK2 Q5S007 2/20 0.38
GSK3B P49841 2/20 0.38
PRKCQ Q04759 2/20 0.38
CHUK O15111 1/20 0.38
PRKD3 O94806 1/20 0.38
CDK1 P06493 1/20 0.38
CDK2 P24941 1/20 0.38
LTK P29376 1/20 0.38
CDK8 P49336 1/20 0.38
PRKX P51817 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15768706 0.85 ROCK2 (0.53) RORCABL1ROCK2ROCK1RPS6KA5
SCHEMBL30282963 0.81 ROCK2 (0.56) ROCK2ROCK1RPS6KA5PKN2LRRK2
Hydrochloric Acid SCHEMBL21640344 0.80 ROCK2 (0.55) ROCK2ROCK1RPS6KA5PKN2LRRK2
SCHEMBL15530710 0.79 PKM (0.53) GSK3BCDK2TP53
Hydrochloric Acid SCHEMBL21640618 0.78 PKM (0.51) GSK3BCDK2TP53
Hydrochloric Acid SCHEMBL30585744 0.78 PKM (0.51) GSK3BCDK2TP53
SCHEMBL19132806 0.76 RORC (0.48) RORCABL1ROCK2ROCK1RPS6KA5
SCHEMBL1554480 0.75 ROCK2 (0.45) RORCABL1ROCK2ROCK1RPS6KA5
SCHEMBL1554477 0.75 ROCK2 (0.45) RORCABL1ROCK2ROCK1RPS6KA5
SCHEMBL2297677 0.74 HPGD (0.62) CLK4TP53TSHRGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2847181-A1 PYRIDAZINE AND PYRIDINE DERIVATIVES AS NAMPT INHIBITORS AbbVie Inc. (US) 2015-03-18 EP claimed
WO-2013170115-A1 PYRIDAZINE AND PYRIDINE DERIVATIVES AS NAMPT INHIBITORS ABBVIE INC. (US) 2013-11-14 WO claimed
EP-2847181-A1 PYRIDAZINE AND PYRIDINE DERIVATIVES AS NAMPT INHIBITORS AbbVie Inc. (US) 2015-03-18 EP disclosed
WO-2013170115-A1 PYRIDAZINE AND PYRIDINE DERIVATIVES AS NAMPT INHIBITORS ABBVIE INC. (US) 2013-11-14 WO disclosed