SCHEMBL15533744

SCHEMBL15533744

COc1ccc(-c2cc(Nc3cccnc3)ncn2)cc1OC

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.61
MAPT P10636 2/20 0.61
KMT2A Q03164 2/20 0.61
CYP1A2 P05177 5/20 0.52
CYP2D6 P10635 5/20 0.52
HSD17B10 Q99714 5/20 0.52
CYP3A4 P08684 4/20 0.52
CLK4 Q9HAZ1 4/20 0.52
CYP2C19 P33261 4/20 0.52
TSHR P16473 2/20 0.52
ABL1 P00519 1/20 0.49
BCR P11274 1/20 0.49
PIK3CD O00329 1/20 0.48
PIK3CA P42336 1/20 0.48
PIK3CG P48736 1/20 0.48
TP53 P04637 2/20 0.47
ALOX15 P16050 2/20 0.47
MAPK1 P28482 2/20 0.47
CHEK1 O14757 1/20 0.47
BACE1 P56817 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4108273 0.82 ALDH1A1 (0.68) CYP1A2CYP2D6HSD17B10CYP3A4CLK4
SCHEMBL15535216 0.79 MAPT (0.49) MEN1MAPTKMT2ACYP1A2CYP2D6
SCHEMBL15533525 0.79 MEN1 (0.62) MEN1MAPTKMT2ACYP1A2CYP2D6
SCHEMBL15533534 0.78 THRB (0.58) MAPTABL1BCRTP53MAPK1
SCHEMBL5923911 0.77 TRPV1 (0.56) MEN1KMT2ACYP1A2CYP2D6HSD17B10
SCHEMBL15533795 0.76 ABL1 (0.64) MEN1MAPTKMT2ACYP1A2CYP2D6
SCHEMBL14742745 0.76 MEN1 (1.00) MEN1MAPTKMT2ACYP1A2MAPK1
SCHEMBL15533662 0.76 CYP2C19 (0.47) MEN1MAPTKMT2ACYP1A2CYP2D6
SCHEMBL27821877 0.76 AHR (0.50) MEN1MAPTKMT2ACYP1A2CYP2D6
SCHEMBL15533812 0.75 ALDH1A1 (0.46) MEN1MAPTKMT2ACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013175415-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND USES THEREOF Piramal Enterprises Limited (IN) 2013-11-28 WO claimed
WO-2013175415-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND USES THEREOF Piramal Enterprises Limited (IN) 2013-11-28 WO disclosed