SCHEMBL15533534

SCHEMBL15533534

COc1ccc(-c2cc(Nc3cccc(C(F)(F)F)c3)ncn2)cc1OC

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.58
ABCG2 Q9UNQ0 4/20 0.55
EGFR P00533 3/20 0.55
ABL1 P00519 6/20 0.54
BCR P11274 6/20 0.54
BRAF P15056 1/20 0.52
TP53 P04637 1/20 0.52
TRPV1 Q8NER1 2/20 0.48
BACE1 P56817 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
ERBB3 P21860 1/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
ERBB4 Q15303 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15533795 0.87 ABL1 (0.64) EGFRABL1BCRTP53TRPV1
SCHEMBL15533950 0.84 ABL1 (0.47) ABCG2ABL1BCRTP53TRPV1
SCHEMBL15533631 0.81 ABL1 (0.46) ABL1BCRBRAFTP53TRPV1
SCHEMBL15533814 0.81 ABL1 (0.59) THRBEGFRABL1BCRBRAF
SCHEMBL15533691 0.80 MAPT (0.47) ABL1BCRTP53NPSR1LMNA
SCHEMBL4237723 0.80 THRB (0.60) THRBABCG2EGFRBRAFTP53
SCHEMBL5923911 0.79 TRPV1 (0.56) EGFRABL1BCRTP53TRPV1
SCHEMBL15534241 0.79 CLK1 (0.63) ABCG2ABL1BCRLMNAMAPT
SCHEMBL15534052 0.79 EGFR (0.55) ABCG2EGFRTP53TRPV1BACE1
SCHEMBL15533744 0.78 MEN1 (0.61) EGFRABL1BCRTP53BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013175415-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND USES THEREOF Piramal Enterprises Limited (IN) 2013-11-28 WO claimed
WO-2013175415-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND USES THEREOF Piramal Enterprises Limited (IN) 2013-11-28 WO disclosed