SCHEMBL1553873

SCHEMBL1553873

CCC(=C(C(=O)O)c1ccncc1)c1cccc(F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.48
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
CYP2C9 P11712 5/20 0.41
CYP1A2 P05177 4/20 0.41
CYP3A4 P08684 4/20 0.41
CYP2D6 P10635 4/20 0.41
CYP2C19 P33261 4/20 0.41
ALDH1A1 P00352 3/20 0.41
HIF1A Q16665 2/20 0.41
TSHR P16473 1/20 0.41
PARP1 P09874 1/20 0.41
LMNA P02545 1/20 0.40
GRM1 Q13255 1/20 0.40
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PLOD2 O00469 1/20 0.40
PLOD3 O60568 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1553870 1.00 KMT2A (0.48) KMT2ACES2CES1CYP2C9CYP1A2
SCHEMBL27555367 0.77 KMT2A (0.49) KMT2ACES2CES1CYP2C9CYP1A2
SCHEMBL1695617 0.76 ESR1 (0.52) KMT2ACYP2C9CYP1A2CYP3A4CYP2D6
SCHEMBL1982008 0.74 CES2 (0.50) CES2CES1SMN1; SMN2
SCHEMBL1982010 0.74 CES2 (0.50) CES2CES1SMN1; SMN2
SCHEMBL3654352 0.73 HTR7 (0.44) KMT2ACES2CES1CYP2C9CYP1A2
SCHEMBL3654354 0.73 HTR7 (0.44) KMT2ACES2CES1CYP2C9CYP1A2
SCHEMBL3654349 0.73 HTR7 (0.44) KMT2ACES2CES1CYP2C9CYP1A2
SCHEMBL3068393 0.73 CES2 (0.74) KMT2ACES2CES1CYP2C9CYP1A2
SCHEMBL1553648 0.71 TP53 (0.48) KMT2ACES2CES1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1439175-B1 PYRIMIDINE COMPOUND AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2011-04-27 EP disclosed