SCHEMBL1554022

SCHEMBL1554022

NC(=O)C(C1CCC(F)(F)CC1)N1CCNCC1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.33
CHRM1 P11229 2/20 0.33
CHRM3 P20309 2/20 0.33
SIGMAR1 Q99720 1/20 0.32
DPP4 P27487 1/20 0.32
DPP7 Q9UHL4 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
CHRNB3 Q05901 1/20 0.32
CHRNA6 Q15825 1/20 0.32
OPRD1 P41143 1/20 0.31
EPHX2 P34913 1/20 0.31
CCR2 P41597 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6187047 0.81 EPHX1 (0.46) CHRM3SIGMAR1DPP4DPP7CHRNB2
SCHEMBL1022186 0.80 CHRNB2 (0.34) SIGMAR1DPP4DPP7CHRNB2CHRNA3
SCHEMBL1022188 0.80 CHRNB2 (0.34) SIGMAR1DPP4DPP7CHRNB2CHRNA3
SCHEMBL1555261 0.78 SIGMAR1 (0.35) CHRM3SIGMAR1CHRNB2CHRNA3CHRNA4
SCHEMBL1554232 0.75 CYP2D6 (0.37) SIGMAR1CHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL1553591 0.75 SIGMAR1 (0.39) SIGMAR1CHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL1555130 0.75 CYP2D6 (0.37) SIGMAR1CHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL6585188 0.73 CPN1 (0.34) DPP4CHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL25380666 0.71 CHRNB2 (0.41) CHRM3SIGMAR1CHRNB2CHRNA3CHRNA4
SCHEMBL978921 0.69 HSD11B1 (0.31) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011000945-A9 AMINOALKAMIDES FOR USE IN THE TREATMENT OF INFLAMMATORY, DEGENERATIVE OR DEMYELINATING DISEASES OF THE CNS NENSIUS RESEARCH A/S (DK) 2011-04-07 WO claimed