SCHEMBL15545458

SCHEMBL15545458

CC(=O)Nc1ccc(C#N)c(S(=O)(=O)C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
ABCC9 O60706 2/20 0.52
ABCC8 Q09428 2/20 0.52
KCNJ11 Q14654 2/20 0.52
KCNJ8 Q15842 2/20 0.52
MAPK1 P28482 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
PLA2G7 Q13093 1/20 0.45
AR P10275 5/20 0.45
CYP2C19 P33261 1/20 0.45
ABCB11 O95342 1/20 0.45
ALB P02768 1/20 0.45
PGR P06401 1/20 0.45
ADRA2C P18825 1/20 0.45
GHSR Q92847 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15606450 0.83 ABCC9 (0.44) ABCC9ABCC8KCNJ11KCNJ8AR
SCHEMBL15606505 0.79 ABCC9 (0.43) ABCC9ABCC8KCNJ11KCNJ8AR
SCHEMBL15544947 0.79 MAPK1 (0.51) ALDH1A1MAPK1SMN1; SMN2
SCHEMBL14289402 0.77 AR (0.59) ALDH1A1PLA2G7ARCYP2C19ABCB11
SCHEMBL15545274 0.76 MEN1 (0.55) ALDH1A1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8351343 0.76 ALDH1A1 (0.79) ALDH1A1SMN1; SMN2PLA2G7CYP2C19
SCHEMBL15545290 0.75 ABCC9 (0.40) ABCC9ABCC8KCNJ11KCNJ8AR
SCHEMBL7057932 0.75 ALDH1A1 (0.63) ALDH1A1SMN1; SMN2PLA2G7CYP2C19
SCHEMBL31125077 0.74 IMPDH2 (0.55) ALDH1A1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL31125117 0.73 KDR (0.55) ARCYP2C19ABCB11ALBPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2870143-B1 TRIAZOLE COMPOUNDS AS ANTIVIRALS HOFFMANN LA ROCHE (CH) 2017-05-17 EP disclosed
EP-2870143-B1 TRIAZOLE COMPOUNDS AS ANTIVIRALS HOFFMANN LA ROCHE (CH) 2017-05-17 EP disclosed
US-20150307461-A1 ANTIVIRAL COMPOUNDS HOFFMANN-LA ROCHE INC. (US) 2015-10-29 US disclosed
US-20150307461-A1 ANTIVIRAL COMPOUNDS HOFFMANN-LA ROCHE INC. (US) 2015-10-29 US disclosed
US-20150307461-A1 ANTIVIRAL COMPOUNDS HOFFMANN-LA ROCHE INC. (US) 2015-10-29 US disclosed
EP-2870143-A1 TRIAZOLE COMPOUNDS AS ANTIVIRALS F. Hoffmann-La Roche AG (CH) 2015-05-13 EP disclosed
US-20140010783-A1 ANTIVIRAL COMPOUNDS HOFFMANN-LA ROCHE INC. 2014-01-09 US disclosed
US-20140010783-A1 ANTIVIRAL COMPOUNDS HOFFMANN-LA ROCHE INC. 2014-01-09 US disclosed
US-20140010783-A1 ANTIVIRAL COMPOUNDS HOFFMANN-LA ROCHE INC. 2014-01-09 US disclosed
WO-2014006066-A1 TRIAZOLE COMPOUNDS AS ANTIVIRALS F. HOFFMANN-LA ROCHE AG (CH) 2014-01-09 WO disclosed
WO-2014006066-A1 TRIAZOLE COMPOUNDS AS ANTIVIRALS F. HOFFMANN-LA ROCHE AG (CH) 2014-01-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150307461-A1 ANTIVIRAL COMPOUNDS HAVCR2, EIF2AK2, MAVS ALDH1A1 222/4885ABCC9 1009/4885ABCC8 1178/4885
US-20140010783-A1 ANTIVIRAL COMPOUNDS HAVCR2, EIF2AK2, MAVS ALDH1A1 222/4885ABCC9 1009/4885ABCC8 1178/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.