SCHEMBL15547835

SCHEMBL15547835

COC1(OC)CCc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.44
MAOB P27338 1/20 0.44
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
SIGMAR1 Q99720 2/20 0.40
TSHR P16473 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
HTR2A P28223 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1820390 0.88 MEN1 (0.51) KDM1AMEN1KMT2ASIGMAR1
SCHEMBL12390025 0.82 MEN1 (0.49) KDM1AMAOBMEN1KMT2ASIGMAR1
SCHEMBL22202531 0.80 SIGMAR1 (0.37) MEN1KMT2ASIGMAR1HTR2A
SCHEMBL10735132 0.79 MEN1 (0.42) KDM1AMAOBMEN1KMT2ASIGMAR1
SCHEMBL2592743 0.78 HTR2A (0.36) MEN1KMT2ASIGMAR1HTR2A
SCHEMBL2468439 0.76 KDM1A (0.46) KDM1AMAOBMEN1KMT2ASIGMAR1
SCHEMBL388323 0.76 KDM1A (0.42) KDM1AMAOBMEN1KMT2ASIGMAR1
SCHEMBL412891 0.76 KDM1A (0.48) KDM1AMAOBMEN1KMT2ATSHR
SCHEMBL29529565 0.76 KDM1A (0.48) KDM1AMAOBMEN1KMT2ATSHR
SCHEMBL6451307 0.75 KDM1A (0.41) KDM1AMAOBMEN1KMT2ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11242344-B2 (4-hydroxypyrrolidin-2-yl)-heterocyclic compounds and methods of use thereof GENENTECH, INC. (US) 2022-02-08 US disclosed
US-20210309660-A1 (4-HYDROXYPYRROLIDIN-2-YL)-HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF GENENTECH INC (US) 2021-10-07 US disclosed
EP-2875362-A1 TEST KIT FOR THE QUANTITATIVE DETERMINATION OF NARCOTIC DRUGS Chiron AS (NO) 2015-05-27 EP disclosed
WO-2014013063-A1 TEST KIT FOR THE QUANTITATIVE DETERMINATION OF NARCOTIC DRUGS CHIRON AS (NO) 2014-01-23 WO disclosed
CN-101772487-B Thyroid compounds TORRENT PHARMACEUTICALS LTD 2014-01-22 CN disclosed
CN-101772487-A Novel compound TORRENT PHARMACEUTICALS LTD 2010-07-07 CN disclosed
CN-101128421-A Methods and compositions for treating amyloid-related diseases NEUROCHEM INTERNAT LTD (CH) 2008-02-20 CN disclosed
CN-1166622-C 2-amino-1, 2-indanes as selective dopamine D3 ligands �������Ŷ���Լ��������˾ 2004-09-15 CN disclosed
CN-1172469-A 2 -aminoindans as selective dopamine D3 ligands UPJOHN CO (US) 1998-02-04 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210309660-A1 (4-HYDROXYPYRROLIDIN-2-YL)-HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF VHL, MDM2, CUL2 KDM1A 1991/4885MAOB 4192/4885MEN1 2547/4885
US-11242344-B2 (4-hydroxypyrrolidin-2-yl)-heterocyclic compounds and methods of use thereof VHL, MDM2, CUL2 KDM1A 1991/4885MAOB 4192/4885MEN1 2547/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.