SCHEMBL15547985

SCHEMBL15547985

O=C(O)N1CCC(C(=O)O)(c2ccnc(Cl)c2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.45
TET3 O43151 4/20 0.45
FBXL19 Q6PCT2 4/20 0.45
CXXC5 Q7LFL8 4/20 0.45
KDM2B Q8NHM5 4/20 0.45
CXXC4 Q9H2H0 4/20 0.45
KDM2A Q9Y2K7 4/20 0.45
TET1 Q8NFU7 3/20 0.42
MEN1 O00255 1/20 0.38
AKR1C3 P42330 2/20 0.36
AKR1C2 P52895 2/20 0.36
AKR1C1 Q04828 2/20 0.36
SMARCA2 P51531 2/20 0.35
SMARCA4 P51532 2/20 0.35
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
APP P05067 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1492751 0.84 AKR1C1 (0.51) KMT2AMEN1AKR1C3AKR1C2AKR1C1
SCHEMBL15535986 0.83 OPRD1 (0.47) KMT2ATET3FBXL19CXXC5KDM2B
SCHEMBL3931269 0.76 KMT2A (0.71) KMT2ATET3FBXL19CXXC5KDM2B
SCHEMBL19029499 0.75 SMARCA2 (0.35) SMARCA2SMARCA4PROKR1
SCHEMBL30872137 0.74 TAS1R3 (0.39) AKR1C3AKR1C2AKR1C1SMARCA2SMARCA4
SCHEMBL23779147 0.74 KMT2A (0.69) KMT2ATET3FBXL19CXXC5KDM2B
SCHEMBL1305563 0.72 KMT2A (0.39) KMT2ATET3FBXL19CXXC5KDM2B
SCHEMBL6179175 0.72 PROKR1 (0.53) KMT2AMEN1AKR1C3PROKR1
SCHEMBL3441871 0.71 ALDH1A1 (0.54) KMT2ATET3FBXL19CXXC5KDM2B
SCHEMBL8514674 0.71 CHRM1 (0.46) KMT2AMEN1AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2852584-A1 SUBSTITUTED DIPYRIDYLAMINES AND USES THEREOF F. Hoffmann-La Roche AG (CH) 2015-04-01 EP disclosed
WO-2013174780-A1 SUBSTITUTED DIPYRIDYLAMINES AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2013-11-28 WO disclosed