SCHEMBL1554920

SCHEMBL1554920

O=CC(c1nc[nH]n1)c1ccc(F)cc1F

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28420380 0.71 IDH1 (0.31) IDO1TDO2
SCHEMBL1515776 0.69 IDO1 (0.51) CES2CES1IDO1TDO2
SCHEMBL28994492 0.67 CES2 (0.38) CES2CES1IDO1TDO2
SCHEMBL3126550 0.66 ALDH1A1 (0.36) CES2CES1IDO1TDO2
SCHEMBL28480587 0.65 CES2 (0.41) CES2CES1IDO1TDO2
SCHEMBL3371037 0.64 CES2 (0.43) CES2CES1IDO1TDO2
SCHEMBL96067 0.64 CES2 (0.43) CES2CES1IDO1TDO2
SCHEMBL1128052 0.64 CES2 (0.43) CES2CES1IDO1TDO2
SCHEMBL7980898 0.64 GABBR2 (0.31)
SCHEMBL5547858 0.63 IDO1 (0.47) CES2CES1IDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011045807-A2 A NOVEL PROCESS TO MANUFACTURE (2R,3S)-2-(2,4-DIFLUOROPHENYL)-3-(5-FLUOROPYRIMIDIN-4-YL)-1-(1H-1,2,4-TRIAZOL-1-YL)BUTAN-2-OL NEULAND LABORATORIES LTD. (IN) 2011-04-21 WO disclosed
EP-0607193-A1 TRIAZOLE ANTIFUNGAL AGENTS Pfizer Limited (GB) 1994-07-27 EP disclosed