SCHEMBL1554939

SCHEMBL1554939

C=C(C)C(=O)OCCC([Si](O[Si](C)(C)C)(O[Si](C)(C)C)O[Si](C)(C)C)([Si](O[Si](C)(C)C)(O[Si](C)(C)C)O[Si](C)(C)C)[Si](O[Si](C)(C)C)(O[Si](C)(C)C)O[Si](C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.43
TSHR P16473 3/20 0.42
ALDH1A1 P00352 2/20 0.38
POLB P06746 1/20 0.33
APEX1 P27695 1/20 0.33
HTT P42858 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
2-Pyrrolidone SCHEMBL9075700 0.83 OR51E2 (0.35) THRBTSHRALDH1A1
SCHEMBL991742 0.82 THRB (0.48) THRBTSHRALDH1A1POLBAPEX1
SCHEMBL6232264 0.79 THRB (0.42) THRBTSHRALDH1A1POLBAPEX1
SCHEMBL396766 0.77 THRB (0.47) THRBTSHRALDH1A1POLBAPEX1
SCHEMBL4454148 0.76 THRB (0.46) THRBTSHRALDH1A1POLBAPEX1
SCHEMBL9302424 0.75 TSHR (0.39) THRBTSHRALDH1A1
SCHEMBL25278638 0.75 THRB (0.44) THRBTSHRALDH1A1POLBAPEX1
SCHEMBL26002227 0.74 THRB (0.55) THRBTSHRALDH1A1POLBAPEX1
SCHEMBL9303996 0.74 THRB (0.47) THRBTSHRALDH1A1POLBAPEX1
SCHEMBL396934 0.74 THRB (0.47) THRBTSHRALDH1A1POLBAPEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9880324-B2 Colored ink for pad transfer printing of silicone hydrogel lenses NOVARTIS AG (CH) 2018-01-30 US disclosed
US-9322960-B2 Method of making a contact lens COOPERVISION INTERNATIONAL HOLDING COMPANY, LP (BB) 2016-04-26 US disclosed
US-9255199-B2 Hydrophilic silicone monomers, process for their preparation and thin films containing the same MOMENTIVE PERFORMANCE MATERIALS INC. (US) 2016-02-09 US disclosed
US-20150247956-A1 METHOD OF MAKING A CONTACT LENS COOPERVISION INTERNATIONAL LIMITED (GB) 2015-09-03 US disclosed
US-9057821-B2 Method of making a contact lens SAUFLON CL LIMITED (GB) 2015-06-16 US disclosed
US-20150076721-A1 COLORED INK FOR PAD TRANSFER PRINTING OF SILICONE HYDROGEL LENSES ALCON INC. (CH) 2015-03-19 US disclosed
US-8920873-B2 Colored ink for pad transfer printing of silicone hydrogel lenses NOVARTIS AG (CH) 2014-12-30 US disclosed
EP-2334382-B1 HYDROPHILIC SILICONE MONOMERS, PROCESS FOR THEIR PREPARATION AND THIN FILMS CONTAINING THE SAME MOMENTIVE PERFORMANCE MAT INC (US) 2014-07-23 EP disclosed
US-20140163135-A1 HYDROPHILIC SILICONE MONOMERS, PROCESS FOR THEIR PREPARATION AND THIN FILMS CONTAINING THE SAME MOMENTIVE PERFORMANCE MATERIALS INC. 2014-06-12 US disclosed
EP-2187243-B1 Colored ink for pad transfer printing of silicone hydrogel lenses NOVARTIS AG (CH) 2012-12-12 EP disclosed
EP-1187873-A1 SURFACE TREATMENT OF SILICONE HYDROGEL CONTACT LENSES COMPRISING HYDROPHILIC POLYMER CHAINS ATTACHED TO AN INTERMEDIATE CARBON COATING BAUSCH & LOMB INCORPORATED (US) 2002-03-20 EP disclosed
EP-1187871-A1 PLASMA SURFACE TREATMENT OF SILICONE HYDROGEL CONTACT LENSES WITH A FLEXIBLE CARBON COATING BAUSCH & LOMB INCORPORATED (US) 2002-03-20 EP disclosed
US-6200626-B1 OXIDATIVE PLASMA TREATMENT; PLASMA POLYMERIZATION; GRAFTING WITH AN ETHYLENICALLY UNSATURATED MONOMER BAUSCH & LOMB INCORPORATED 2001-03-13 US disclosed
WO-2000071611-A1 PLASMA SURFACE TREATMENT OF SILICONE HYDROGEL CONTACT LENSES WITH A FLEXIBLE CARBON COATING BAUSCH & LOMB INCORPORATED (US) 2000-11-30 WO disclosed
WO-2000071613-A1 SURFACE TREATMENT OF SILICONE HYDROGEL CONTACT LENSES COMPRISING HYDROPHILIC POLYMER CHAINS ATTACHED TO AN INTERMEDIATE CARBON COATING BAUSCH & LOMB INCORPORATED (US) 2000-11-30 WO disclosed
WO-2000071612-A1 SURFACE-TREATMENT OF SILICONE MEDICAL DEVICES COMPRISING AN INTERMEDIATE CARBON COATING AND GRAFT POLYMERIZATION BAUSCH & LOMB INCORPORATED (US) 2000-11-30 WO disclosed
EP-0652823-A1 PROCESS FOR MAKING SILICONE CONTAINING HYDROGEL LENSES BAUSCH & LOMB INCORPORATED (US) 1995-05-17 EP disclosed
US-5346976-A Itaconate copolymeric compositions for contact lenses POLYMER TECHNOLOGY CORPORATION (US) 1994-09-13 US disclosed
WO-1994003324-A1 PROCESS FOR MAKING SILICONE CONTAINING HYDROGEL LENSES BAUSCH & LOMB INCORPORATED (US) 1994-02-17 WO disclosed
EP-0277771-A2 Continuous-wear lenses having improved physical properties BAUSCH & LOMB INCORPORATED (US) 1988-08-10 EP disclosed