SCHEMBL15566852

SCHEMBL15566852

Fc1ccc(F)c([C]2CC2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 2/20 0.42
CA3 P07451 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42
CA14 Q9ULX7 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
PTPN1 P18031 1/20 0.39
PARP1 P09874 1/20 0.38
PARP10 Q53GL7 1/20 0.38
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
KDM1A O60341 2/20 0.38
KDM1B Q8NB78 1/20 0.38
ALDH1A1 P00352 2/20 0.37
IDH1 O75874 1/20 0.37
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
THRB P10828 1/20 0.35
HK1 P19367 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28289816 0.91 CA9 (0.39) CA9CA3CA6CA5ACA14
SCHEMBL9766850 0.81 CA9 (0.52) CA9CA3CA6CA5ACA14
SCHEMBL434353 0.80 ALDH1A1 (0.42) CA9CA3CA6CA5ACA14
SCHEMBL6901382 0.73 MPL (0.47) PARP1PARP10KDM1ACYP11B1CYP11B2
SCHEMBL24766983 0.72 CA3 (0.44) CA9CA3CA6CA5ACA14
SCHEMBL21408274 0.72 ERN1 (0.45) KDM4ENFE2L2
SCHEMBL435076 0.71 ALDH1A1 (0.39) CA9CA3CA6CA5ACA14
SCHEMBL436723 0.71 MAOA (0.41) CES2CES1ALDH1A1KDM4ELMNA
SCHEMBL30927149 0.71 ALDH1A1 (0.50) CA9CA3CA6CA5ACA14
SCHEMBL3019057 0.71 PTGS2 (0.44) ACHECYP19A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2882722-A1 QUINOXALINE DERIVATIVES AS GPR6 MODULATORS Envoy Therapeutics Inc. (US) 2015-06-17 EP disclosed
WO-2014028479-A1 QUINOXALINE DERIVATIVES AS GPR6 MODULATORS ENVOY THERAPEUTICS, INC. (US) 2014-02-20 WO disclosed