SCHEMBL15568178

SCHEMBL15568178

O=C(O)c1ccc(-c2nc3ccccc3n2Cc2ccccc2)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.74
PDE6D O43924 2/20 0.74
ALDH2 P05091 1/20 0.74
ALDH3A1 P30838 1/20 0.74
PIN1 Q13526 5/20 0.66
TP53 P04637 4/20 0.64
MAPT P10636 2/20 0.64
HTT P42858 2/20 0.64
SMN1; SMN2 Q16637 2/20 0.64
HPGD P15428 1/20 0.64
NPSR1 Q6W5P4 1/20 0.64
DRD2 P14416 1/20 0.64
TBXA2R P21731 1/20 0.64
PPARG P37231 1/20 0.63
AGTR1 P30556 2/20 0.60
AGTR2 P50052 2/20 0.60
BRD4 O60885 1/20 0.60
KDM4E B2RXH2 2/20 0.59
LMNA P02545 1/20 0.59
CNR2 P34972 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2884309 0.95 ALDH1A1 (0.74) ALDH1A1PDE6DALDH2ALDH3A1PIN1
SCHEMBL29056606 0.86 ALDH1A1 (0.65) ALDH1A1PDE6DALDH2ALDH3A1PIN1
SCHEMBL15568695 0.86 TP53 (0.70) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL229828 0.85 ALDH1A1 (1.00) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL28503579 0.85 ALDH1A1 (0.63) ALDH1A1PDE6DALDH2ALDH3A1PIN1
SCHEMBL28503563 0.85 ALDH1A1 (0.63) ALDH1A1PDE6DALDH2ALDH3A1PIN1
SCHEMBL15567152 0.85 ALDH1A1 (0.72) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL15474496 0.85 ALDH1A1 (0.80) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL15569395 0.83 ALDH1A1 (0.78) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL5010971 0.83 ALDH1A1 (1.00) ALDH1A1PDE6DALDH2ALDH3A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO claimed
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO disclosed