SCHEMBL28503579

SCHEMBL28503579

O=C(O)c1ccc2nc(-c3ccccc3)n(Cc3ccccc3)c2c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.63
PDE6D O43924 2/20 0.63
ALDH2 P05091 1/20 0.63
ALDH3A1 P30838 1/20 0.63
RHEB Q15382 1/20 0.59
BRD4 O60885 3/20 0.57
TP53 P04637 4/20 0.55
MAPT P10636 2/20 0.54
CYP11B2 P19099 1/20 0.54
SMN1; SMN2 Q16637 2/20 0.52
LMNA P02545 1/20 0.52
RECQL P46063 1/20 0.52
RAB9A P51151 1/20 0.52
DRD2 P14416 1/20 0.51
TBXA2R P21731 1/20 0.51
HPGD P15428 1/20 0.50
HTT P42858 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
PIN1 Q13526 1/20 0.50
HDAC1 Q13547 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28503563 0.90 ALDH1A1 (0.63) ALDH1A1PDE6DALDH2ALDH3A1RHEB
SCHEMBL28505411 0.87 DRD2 (0.66) ALDH1A1PDE6DALDH2ALDH3A1BRD4
SCHEMBL14382294 0.86 PDE2A (0.61) ALDH1A1PDE6DALDH2ALDH3A1BRD4
SCHEMBL15568178 0.85 ALDH1A1 (0.74) ALDH1A1PDE6DALDH2ALDH3A1BRD4
SCHEMBL6169195 0.85 TNF (0.62) BRD4RAB9AHDAC1HDAC6HSD17B10
SCHEMBL2884309 0.85 ALDH1A1 (0.74) ALDH1A1PDE6DALDH2ALDH3A1RHEB
SCHEMBL15568695 0.85 TP53 (0.70) ALDH1A1PDE6DALDH2ALDH3A1BRD4
SCHEMBL6170384 0.84 HDAC1 (0.57) ALDH1A1RHEBMAPTRAB9AHDAC1
SCHEMBL6475293 0.82 ALDH1A1 (0.68) ALDH1A1PDE6DALDH2ALDH3A1BRD4
SCHEMBL28508255 0.82 BRD4 (0.52) ALDH1A1PDE6DALDH2ALDH3A1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107311933-B Benzimidazole derivative, preparation method and application thereof 中国人民解放军军事医学科学院毒物药物研究所 2020-12-22 CN disclosed