SCHEMBL28503563

SCHEMBL28503563

O=C(O)c1ccc2c(c1)nc(-c1ccccc1)n2Cc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.63
PDE6D O43924 2/20 0.63
ALDH2 P05091 1/20 0.63
ALDH3A1 P30838 1/20 0.63
JAK2 O60674 2/20 0.59
JAK1 P23458 2/20 0.59
TYK2 P29597 2/20 0.59
JAK3 P52333 2/20 0.59
RHEB Q15382 1/20 0.59
TP53 P04637 4/20 0.55
HCAR3 P49019 1/20 0.55
MAPT P10636 2/20 0.54
PTGER4 P35408 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.52
LMNA P02545 1/20 0.52
RECQL P46063 1/20 0.52
RAB9A P51151 1/20 0.52
HTT P42858 2/20 0.52
DRD2 P14416 1/20 0.51
TBXA2R P21731 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28503579 0.90 ALDH1A1 (0.63) ALDH1A1PDE6DALDH2ALDH3A1RHEB
SCHEMBL2884309 0.85 ALDH1A1 (0.74) ALDH1A1PDE6DALDH2ALDH3A1RHEB
SCHEMBL15568178 0.85 ALDH1A1 (0.74) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL15568695 0.85 TP53 (0.70) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL9662852 0.83 PTGER4 (0.66) ALDH1A1JAK2JAK1TYK2JAK3
SCHEMBL28507437 0.82 PTGER4 (0.55) ALDH1A1PDE6DALDH2ALDH3A1JAK2
SCHEMBL8233038 0.81 NLRP3 (0.74) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL594322 0.80 ALDH1A1 (0.68) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL28547289 0.80 ALDH1A1 (0.60) ALDH1A1PDE6DALDH2ALDH3A1TP53
SCHEMBL6171734 0.79 PPARG (0.66)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107311933-B Benzimidazole derivative, preparation method and application thereof 中国人民解放军军事医学科学院毒物药物研究所 2020-12-22 CN disclosed