D-Glutamate

D-Glutamate

SCHEMBL15577173

CC(O)C(=O)O.CC(O)C(=O)O.C[N+](C)(C)CCO.NC(CCC(=O)O)C(=O)[O-]

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3GNRHRMPLPDE3APDE3BPDE4APDE4BPDE4CPDE4DPPARASLC5A2

The experimentally established mechanism targets of D-Glutamate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.43
GRM8 O00222 1/20 0.43
GRM6 O15303 1/20 0.43
GRIN2D O15399 1/20 0.43
GRIN3B O60391 1/20 0.43
GSR P00390 1/20 0.43
GRIK1 P39086 1/20 0.43
GRM5 P41594 1/20 0.43
GRIA1 P42261 1/20 0.43
GRIA2 P42262 1/20 0.43
GRIA3 P42263 1/20 0.43
SLC1A3 P43003 1/20 0.43
SLC1A2 P43004 1/20 0.43
SLC1A1 P43005 1/20 0.43
GRIA4 P48058 1/20 0.43
GRIN1 Q05586 1/20 0.43
GRIN2A Q12879 1/20 0.43
GRIK2 Q13002 1/20 0.43
GRIK3 Q13003 1/20 0.43
GRIN2B Q13224 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
D-Glutamate SCHEMBL8218834 0.93 CYP1A2 (0.46) CYP1A2GRM8GRM6GRIN2DGRIN3B
Glutamic Acid SCHEMBL15577174 0.91 CYP1A2 (0.51) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL10623300 0.83 GRM8 (0.64) CYP1A2GRM8GRM6GRIN2DGRIN3B
Glutamic Acid SCHEMBL10623303 0.83 GRM8 (0.64) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL28219176 0.82 GRM8 (0.62) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL15577133 0.82 BBOX1 (0.43) LMNAKMT2AMEN1CYP3A4SLC5A7
D-Glutamate SCHEMBL8218829 0.82 BBOX1 (0.43) LMNAKMT2AMEN1CYP3A4SLC5A7
D-Glutamate SCHEMBL16241512 0.80 CYP1A2 (0.57) CYP1A2GRM8GRM6GRIN2DGRIN3B
Choline SCHEMBL3820379 0.78 MEN1 (0.55) LMNAKMT2AMEN1MAPTCYP3A4
Aspartic Acid SCHEMBL6033509 0.77 LMNA (0.41) LMNAKMT2AMEN1MAPTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2895071-A1 ROD SHAPED IMPLANTABLE BIOSENSOR Brains Online Holding B.V. (NL) 2015-07-22 EP disclosed
WO-2014041190-A1 ROD SHAPED IMPLANTABLE BIOSENSOR BRAINS ONLINE HOLDING B.V. (NL) 2014-03-20 WO disclosed