SCHEMBL15577253

SCHEMBL15577253

OCCC1(c2ccccc2)CCCOC1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.43
CYP2D6 P10635 2/20 0.41
EPHX2 P34913 1/20 0.41
SLC6A4 P31645 6/20 0.39
SLC6A2 P23975 6/20 0.39
SLC6A3 Q01959 6/20 0.39
LMNA P02545 2/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
MAPK1 P28482 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
S1PR1 P21453 1/20 0.36
S1PR3 Q99500 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29017348 0.87 DPP4 (0.46) DPP4SLC6A4SLC6A2SLC6A3LMNA
SCHEMBL29017424 0.87 DPP4 (0.46) DPP4SLC6A4SLC6A2SLC6A3LMNA
SCHEMBL3380377 0.83 ACSS2 (0.43) DPP4CYP2D6EPHX2SLC6A4SLC6A2
SCHEMBL29017350 0.81 ICMT (0.39) DPP4CYP2D6EPHX2MAOAMAOB
SCHEMBL18440465 0.81 DPP4 (0.53) DPP4CYP2D6EPHX2SLC6A4SLC6A2
SCHEMBL15577241 0.80 ICMT (0.51) DPP4LMNAMAOAMAOBTAAR1
SCHEMBL15577265 0.79 TSHR (0.54) DPP4EPHX2LMNAMEN1KMT2A
SCHEMBL24641080 0.77 MAOA (0.42) DPP4SLC6A4SLC6A2SLC6A3LMNA
SCHEMBL1124803 0.77 MAOA (0.56) DPP4CYP2D6EPHX2SLC6A4SLC6A2
SCHEMBL29017375 0.76 MAOA (0.42) DPP4MAOAMAOBTAAR1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014041349-A1 TETRAHYDROPYRAN-4-YLETHYLAMINO- OR TETRAHYDROPYRANYL-4-ETHYLOXY-PYRIMIDINES OR -PYRIDAZINES AS ISOPRENYLCYSTEINCARBOXYMETHYL TRANSFERASE INHIBITORS CANCER THERAPEUTICS CRC PTY LTD (AU) 2014-03-20 WO disclosed