SCHEMBL15580700

SCHEMBL15580700

COC(=O)c1cnc(Oc2ccc([C@@H](C)[C@@](O)(c3ccc4oc(=O)n(C)c4c3)C(C)(F)F)c(Cl)c2)nc1

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.32
GPR55 Q9Y2T6 2/20 0.32
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
P2RX3 P56373 1/20 0.31
LMNA P02545 1/20 0.31
PDK1 Q15118 2/20 0.31
PDK2 Q15119 2/20 0.31
PDK3 Q15120 2/20 0.31
PDK4 Q16654 2/20 0.31
LRRK2 Q5S007 1/20 0.31
KDR P35968 3/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12164236 0.95 MET (0.32) METGPR55ALDH1A1TSHRP2RX3
SCHEMBL473920 0.95 MET (0.32) METGPR55ALDH1A1TSHRP2RX3
SCHEMBL12164237 0.87 PTGER4 (0.33) GPR55LRRK2
SCHEMBL473996 0.87 PTGER4 (0.33) GPR55LRRK2
SCHEMBL15520201 0.87 GPR55 (0.32) GPR55LMNALRRK2MEN1KMT2A
SCHEMBL473965 0.86 LMNA (0.34) METGPR55ALDH1A1TSHRP2RX3
SCHEMBL12164178 0.86 LMNA (0.41) METALDH1A1TSHRP2RX3LMNA
SCHEMBL12164179 0.86 LMNA (0.34) METGPR55ALDH1A1TSHRP2RX3
SCHEMBL473932 0.86 LMNA (0.41) METALDH1A1TSHRP2RX3LMNA
SCHEMBL15519897 0.84 KMO (0.32) GPR55LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP disclosed