SCHEMBL15580925

SCHEMBL15580925

CC(=O)[15NH]c1cccc2c1C(=O)OC2=O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.61
ALDH1A1 P00352 3/20 0.59
KDM4E B2RXH2 2/20 0.59
HPGD P15428 2/20 0.59
GAA P10253 1/20 0.59
HSD17B10 Q99714 1/20 0.59
CASP3 P42574 1/20 0.56
AHR P35869 1/20 0.50
CCNE2 O96020 9/20 0.49
CCNE1 P24864 9/20 0.49
CDK2 P24941 9/20 0.49
SMN1; SMN2 Q16637 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
DDB1 Q16531 1/20 0.45
CRBN Q96SW2 1/20 0.45
CDK4 P11802 4/20 0.45
CCND1 P24385 4/20 0.45
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL303302 1.00 MAOA (0.61) MAOAALDH1A1KDM4EHPGDGAA
SCHEMBL29860722 1.00 MAOA (0.61) MAOAALDH1A1KDM4EHPGDGAA
SCHEMBL705018 0.89 MAOA (0.49) MAOAALDH1A1KDM4EHPGDGAA
SCHEMBL17580121 0.89 MAOA (0.49) MAOAALDH1A1KDM4EHPGDGAA
SCHEMBL17590085 0.85 MAOA (0.44) MAOAALDH1A1KDM4EHPGDGAA
SCHEMBL3828974 0.83 MAOA (0.51) MAOAALDH1A1KDM4EHPGDGAA
SCHEMBL15444503 0.83 MAOA (0.43) MAOAALDH1A1KDM4EHPGDGAA
SCHEMBL18328582 0.83 CA1 (0.43) MAOAALDH1A1KDM4EHPGDGAA
SCHEMBL20334273 0.80 MAOA (0.90) MAOAALDH1A1KDM4EHPGDGAA
SCHEMBL29986841 0.79 MAOA (0.87) MAOAALDH1A1KDM4EHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9642836-B2 Isotopologues of isoindole derivatives CELGENE CORPORATION (US) 2017-05-09 US disclosed
US-20150258063-A1 ISOTOPOLOGUES OF ISOINDOLE DERIVATIVES AMGEN INC. 2015-09-17 US disclosed
US-9045417-B2 Isotopologues of isoindole derivatives CELGENE CORPORATION (US) 2015-06-02 US disclosed
US-8981117-B2 Processes for the preparation of isoindole compounds and isotopologues thereof CELGENE CORPORATION (US) 2015-03-17 US disclosed
US-20140194485-A1 ISOTOPOLOGUES OF ISOINDOLE DERIVATIVES CELGENE CORPORATION (US) 2014-07-10 US disclosed
US-20140081032-A1 PROCESSES FOR THE PREPARATION OF ISOINDOLE COMPOUNDS AND ISOTOPOLOGUES THEREOF CELGENE CORPORATION (US) 2014-03-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140081032-A1 PROCESSES FOR THE PREPARATION OF ISOINDOLE COMPOUNDS AND ISOTOPOLOGUES THEREOF HPD, DHPS, IDH2 MAOA 916/4885ALDH1A1 1488/4885KDM4E 2320/4885
US-20140194485-A1 ISOTOPOLOGUES OF ISOINDOLE DERIVATIVES IDO1, CYP11B2, IDO2 MAOA 556/4885ALDH1A1 1321/4885KDM4E 2562/4885
US-20150258063-A1 ISOTOPOLOGUES OF ISOINDOLE DERIVATIVES IDO1, CYP11B2, IDO2 MAOA 556/4885ALDH1A1 1321/4885KDM4E 2562/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.