SCHEMBL15616400

SCHEMBL15616400

O=C(NC1CCC(O)CC1)c1ccc(Cl)c(-c2ccc3c(c2)CCCN3)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 8/20 0.53
RORC P51449 1/20 0.47
KDM4E B2RXH2 1/20 0.46
MAPT P10636 1/20 0.46
RIPK2 O43353 2/20 0.44
CHEK1 O14757 3/20 0.43
SGK1 O00141 1/20 0.42
AURKA O14965 1/20 0.42
CSNK2A2 P19784 1/20 0.42
AKT1 P31749 1/20 0.42
AKT2 P31751 1/20 0.42
CSNK2B P67870 1/20 0.42
CSNK2A1 P68400 1/20 0.42
AKT3 Q9Y243 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
SMYD3 Q9H7B4 3/20 0.41
RAF1 P04049 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL45469 0.82 KDM4E (0.67) KDM4EMAPTHDAC8SMYD3
SCHEMBL45245 0.78 KDM4E (0.65) KDM4EMAPTHDAC8SMYD3
SCHEMBL16061494 0.74 KDM4E (0.59) KDM4EMAPTHDAC8SMYD3
SCHEMBL15616643 0.73 ALDH1A1 (0.47) RORCKDM4EMAPT
SCHEMBL15616410 0.72 RORC (0.89) RORC
SCHEMBL45293 0.72 KDM4E (0.62) KDM4EMAPTHDAC8SMYD3
SCHEMBL15616523 0.72 PPARG (0.51) MAPT
SCHEMBL3200151 0.71 NPC1 (0.68) MAPK14KDM4EMAPTRIPK2SMYD3
SCHEMBL3211244 0.69 MAPK14 (0.62) MAPK14RORCRIPK2SMYD3
SCHEMBL1232193 0.69 MAPK14 (1.00) MAPK14RAF1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014008214-A1 BIARYL-CONTAINING COMPOUNDS AS INVERSE AGONISTS OF ROR-GAMMA RECEPTORS BIOGEN IDEC MA INC. (US) 2014-01-09 WO disclosed