SCHEMBL1561876

SCHEMBL1561876

CN1CCN(C(=O)N(C)C2CC#CCC2)CC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.40
HSD11B1 P28845 1/20 0.37
VNN1 O95497 1/20 0.37
CYP1A2 P05177 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
EPHX2 P34913 1/20 0.35
HTT P42858 2/20 0.34
ALDH1A1 P00352 3/20 0.34
LMNA P02545 2/20 0.33
MCHR1 Q99705 1/20 0.32
KDM4E B2RXH2 2/20 0.31
MAPT P10636 1/20 0.31
ALOX15 P16050 1/20 0.31
TSHR P16473 1/20 0.31
PPP5C P53041 2/20 0.31
PPP2CA P67775 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1562085 0.84 CHRNB2 (0.38) HSD11B1EPHX2MCHR1
SCHEMBL1562092 0.84 MAPT (0.44) VNN1CYP1A2MAPTTSHR
SCHEMBL18389969 0.80 HTR1A (0.50) HTR1AHSD11B1VNN1CYP1A2TDP1
SCHEMBL25568891 0.79 HTR1A (0.48) HTR1AHSD11B1VNN1CYP1A2TDP1
SCHEMBL1561215 0.76 LMNA (0.49) HTR1AHSD11B1VNN1CYP1A2TDP1
SCHEMBL1561751 0.73
SCHEMBL1561145 0.73 HTR1A (0.43) HTR1AHSD11B1VNN1CYP1A2TDP1
SCHEMBL19012442 0.73 MAPT (0.45) HTR1AHSD11B1VNN1CYP1A2TDP1
SCHEMBL1561358 0.72
SCHEMBL24371412 0.71 VNN1 (0.50) HTR1AVNN1CYP1A2TDP1MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091925-B1 BICYCLIC HETEROCYCLES, MEDICAMENTS CONTAINING SAID COMPOUNDS, USE THEREOF, AND METHOD FOR PRODUCTION OF SAME BOEHRINGER INGELHEIM INT (DE) 2011-04-06 EP claimed