SCHEMBL156197

SCHEMBL156197

[c]1ccc2c(n1)CCCC2

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.35
ADRA2B P18089 2/20 0.35
ADRA2C P18825 2/20 0.35
TSHR P16473 1/20 0.35
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
SIGMAR1 Q99720 1/20 0.32
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17986607 0.98 ADRA2A (0.34) ADRA2AADRA2BADRA2CTSHRHTR2A
SCHEMBL338410 0.98 ADRA2A (0.34) ADRA2AADRA2BADRA2CTSHRHTR2A
SCHEMBL569626 0.95
SCHEMBL4986870 0.77 HTR2C (0.41) HTR2AHTR2C
SCHEMBL1827327 0.71 PDK1 (0.30)
SCHEMBL223932 0.71 PNMT (0.41) ADRA2AADRA2BADRA2CHTR2AHTR2C
SCHEMBL1834181 0.69
SCHEMBL21591664 0.69 MAOA (0.46) ADRA2A
SCHEMBL20723049 0.69 PLAU (0.44)
SCHEMBL1834182 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6531 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118344342-A Substituted polyaromatic ring derivatives, compositions and uses thereof 康迈迪森(北京)医药科技有限公司 2024-07-16 CN claimed
CN-118324816-A Organometallic compound, light-emitting device, electronic apparatus, and electronic device 三星显示有限公司 2024-07-12 CN claimed
US-11987588-B2 Modulators of the beta-3 adrenergic receptor useful for the treatment or prevention of heart failure and disorders related thereto ARENA PHARMACEUTICALS, INC. (US) 2024-05-21 US claimed
CN-117917420-A Organometallic compound, light-emitting device, electronic apparatus, and electronic device 三星显示有限公司 2024-04-23 CN claimed
EP-4353262-A1 NOVEL COMPOUND HAVING INHIBITORY ACTIVITY AGAINST PENDRIN, AND PHARMACEUTICAL USES THEREOF UIF (University Industry Foundation), Yonsei University (KR) 2024-04-17 EP claimed
CN-117529202-A Organometallic compound, light-emitting device, electronic apparatus, and electronic device 三星显示有限公司 2024-02-06 CN claimed
CN-117135987-A Organometallic compound, light-emitting device including the same, electronic device, and electronic device 三星显示有限公司 2023-11-28 CN claimed
CN-109411632-B Organic light emitting device and apparatus including the same 三星显示有限公司 2023-11-24 CN claimed
CN-117062455-A Organic light emitting device and electronic apparatus including the same 三星显示有限公司 2023-11-14 CN claimed
US-20230278958-A1 TRICYCLIC HETEROCYCLES MERCK PATENT GMBH (DE) 2023-09-07 US claimed
US-4831026-A ANTIBIOTICS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1989-05-16 US claimed
EP-0215435-A1 2-Oxa-isocephem compounds, compositions containing same and processes for preparing same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1987-03-25 EP claimed
US-4639519-A 2-substituted alkylaminopyrimidones useful as H2 -antagonists and antiinflamatory agents SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1987-01-27 US claimed
US-4558128-A ANTIHISTAMINE, ANTIINFLAMMATORY AGENT SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1985-12-10 US claimed
US-4523015-A Process and nitroaminopyrimidone intermediates for histamine H2 -antagonists SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1985-06-11 US claimed
US-4496567-A HSITAMINE H2 ANTAGONISTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1985-01-29 US claimed
EP-0013071-B1 PYRIMIDINONE DERIVATIVES, PROCESSES FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1983-11-16 EP claimed
US-4305945-A Isoureas and isothioureas SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1981-12-15 US claimed
EP-0003677-B1 PYRIMIDONES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1981-11-11 EP claimed
EP-0003677-A2 Pyrimidones, processes for their preparation and pharmaceutical compositions containing them SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1979-08-22 EP claimed