SCHEMBL15624596

SCHEMBL15624596

COc1cccc(-c2scnc2N)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.41
RIPK2 O43353 2/20 0.38
IRAK4 Q9NWZ3 1/20 0.36
ALOX5AP P20292 1/20 0.36
KDR P35968 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA3 P34903 1/20 0.36
TAAR1 Q96RJ0 1/20 0.35
MAP4K4 O95819 1/20 0.35
IDH1 O75874 1/20 0.35
TRPV4 Q9HBA0 1/20 0.35
TGFBR1 P36897 1/20 0.35
HASPIN Q8TF76 1/20 0.35
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
RAB9A P51151 1/20 0.34
BACE1 P56817 1/20 0.34
PDE10A Q9Y233 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10304995 0.84 BTK (0.41) BTKRIPK2IRAK4ALOX5APKDR
SCHEMBL15624594 0.77 CYP11B2 (0.37) BACE1
SCHEMBL3155981 0.74 BTK (0.61) BTKKDRGABRA1GABRG2GABRB3
SCHEMBL21484628 0.73 ALDH1A1 (0.51) BTKNPC1ALDH1A1RAB9A
SCHEMBL13745852 0.71 BTK (0.41) BTKALOX5APGABRA1GABRG2GABRB3
SCHEMBL2184656 0.69 RAB9A (0.49) BTKRAB9A
SCHEMBL15692562 0.68 KDM4E (0.50) TGFBR1NPC1ALDH1A1RAB9APDE10A
SCHEMBL25902083 0.68 BTK (0.41) BTKALOX5APIDH1TGFBR1
SCHEMBL160602 0.67 BTK (0.47) BTKKDRNPC1ALDH1A1RAB9A
SCHEMBL25027832 0.67 BTK (0.46) BTKKDRGABRA1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2252595-B1 OXIM DERIVATIVES AS HSP90 INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2014-03-26 EP disclosed