SCHEMBL15633889

SCHEMBL15633889

CC1(C)CCC(N(CCOc2ccc(-c3cccc(-n4cc[nH]c4=O)c3)cc2)C(=O)O)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CPT2 P23786 1/20 0.41
CPT1A P50416 1/20 0.41
CPT1B Q92523 1/20 0.41
PPARD Q03181 2/20 0.33
PPARA Q07869 1/20 0.33
MCHR1 Q99705 3/20 0.33
KCNH2 Q12809 1/20 0.33
PDE3B Q13370 3/20 0.32
PDE3A Q14432 3/20 0.32
P2RY12 Q9H244 3/20 0.32
HRH3 Q9Y5N1 2/20 0.32
CYP2D6 P10635 1/20 0.32
SLC9A3 P48764 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 3/20 0.32
TP53 P04637 2/20 0.32
PDE2A O00408 2/20 0.32
LMNA P02545 1/20 0.32
FFAR4 Q5NUL3 1/20 0.32
ADAMTS5 Q9UNA0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12651138 0.90 CPT2 (0.39) CPT2CPT1ACPT1BPPARDPPARA
SCHEMBL1788720 0.82 ALDH1A1 (0.40) CPT2CPT1ACPT1BHRH3CYP2D6
Hydrochloric Acid SCHEMBL3339930 0.81 ALDH1A1 (0.40) CPT2CPT1ACPT1BHRH3CYP2D6
SCHEMBL15633618 0.79 CPT1A (0.36) CPT1AKCNH2HRH3ALDH1A1MAPT
SCHEMBL3338423 0.78 HRH2 (0.46) PPARAMCHR1FFAR4
SCHEMBL15634006 0.75 KIF11 (0.41) CPT2CPT1AMCHR1KCNH2ALDH1A1
SCHEMBL3338354 0.75 FFAR4 (0.35) PPARDPPARAMCHR1ALDH1A1FFAR4
SCHEMBL3368490 0.72 ALDH1A1 (0.45) MCHR1HRH3ALDH1A1MAPTLMNA
SCHEMBL12607437 0.71 CYP1A2 (0.39) KCNH2PDE3BPDE3AHRH3CYP2D6
SCHEMBL12607465 0.70 MAPT (0.41) CPT1ASLC9A3MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8822518-B2 Compounds as antagonists or inverse agonists of opioid receptors for treatment of addiction GLAXOSMITHKLINE LLC (US) 2014-09-02 US disclosed
US-20140100255-A1 Novel Compounds As Antagonists Or Inverse Agonists At Opioid Receptors GLAXOSMITHKLINE LLC (US) 2014-04-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140100255-A1 Novel Compounds As Antagonists Or Inverse Agonists At Opioid Receptors OPRL1, OPRM1, OPRK1 CPT2 3231/4885CPT1A 1309/4885CPT1B 2238/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.