SCHEMBL15705331

SCHEMBL15705331

NC(O)c1ccccc1C(N)Cc1ccncc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
SLC6A4 P31645 2/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A3 Q01959 1/20 0.41
ALPI P09923 1/20 0.38
PKM P14618 1/20 0.38
PTGS1 P23219 1/20 0.38
XIAP P98170 1/20 0.38
SLC7A5 Q01650 1/20 0.38
ALDH1A1 P00352 1/20 0.37
ANPEP P15144 1/20 0.36
ERAP2 Q6P179 1/20 0.36
ERAP1 Q9NZ08 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.36
EPHX1 P07099 1/20 0.35
ROCK2 O75116 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1156871 0.79 SLC6A4 (0.41) CYP3A4CYP1A2CYP2C9CYP2C19SLC6A4
SCHEMBL1157043 0.74 SLC6A4 (0.60) CYP1A2CYP2C19SLC6A4SLC6A2SLC6A3
SCHEMBL1157137 0.73 CYP1A2 (0.47) CYP3A4CYP1A2CYP2C9CYP2C19SLC6A4
Hydrochloric Acid SCHEMBL9322405 0.73 SLC6A4 (0.58) SLC6A4SLC6A2SLC6A3EPHX1CYP2D6
Hydrochloric Acid SCHEMBL9322527 0.73 SLC6A4 (0.58) SLC6A4SLC6A2SLC6A3EPHX1CYP2D6
SCHEMBL6765024 0.72 LMNA (0.40) CYP3A4CYP1A2SLC6A2ALPIPKM
SCHEMBL9306936 0.71 DPP4 (0.55) CYP3A4CYP1A2CYP2C9CYP2C19SLC6A4
SCHEMBL8867023 0.71 SLC6A2 (0.66) CYP1A2SLC6A4SLC6A2SLC6A3ANPEP
SCHEMBL6890878 0.70 GRIN2D (0.42) CYP3A4CYP1A2SLC6A4SLC6A2SLC6A3
SCHEMBL19143563 0.70 CYP3A4 (0.52) CYP3A4CYP1A2CYP2C9CYP2C19SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140128352-A1 COMPOUNDS AND METHODS FOR MODULATING MITOCHONDRIAL METABOLISM AND REACTIVE OXYGEN SPECIES PRODUCTION BUCK INSTITUTE FOR RESEARCH ON AGING (US) 2014-05-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140128352-A1 COMPOUNDS AND METHODS FOR MODULATING MITOCHONDRIAL METABOLISM AND REACTIVE OXYGEN SPECIES PRODUCTION PC, PCK2, TXNRD2 CYP3A4 368/4885CYP1A2 480/4885CYP2C9 967/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.