SCHEMBL1573474

SCHEMBL1573474

COc1cccc(CN(C)C(=O)C(Sc2ccccc2)c2cc(OC)cc(OC)c2)c1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.51
MEN1 O00255 5/20 0.48
KMT2A Q03164 5/20 0.48
HSD17B2 P37059 5/20 0.47
POLB P06746 1/20 0.43
HPGD P15428 1/20 0.43
RECQL P46063 1/20 0.43
CALM1 P0DP23 1/20 0.43
CAMKK2 Q96RR4 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TSPO P30536 1/20 0.43
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1573360 0.91 MEN1 (0.46) TACR1MEN1KMT2AHSD17B2POLB
SCHEMBL1573013 0.77 TACR1 (0.49) TACR1MEN1KMT2AHSD17B2POLB
SCHEMBL15831230 0.76 MEN1 (0.62) MEN1KMT2AHSD17B2POLBHPGD
SCHEMBL1572940 0.76 LMNA (0.51) TACR1MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL9112410 0.74 TACR1 (0.70) TACR1MEN1KMT2AHPGDALDH1A1
SCHEMBL10702424 0.73 MAPT (0.55) ALDH1A1SMN1; SMN2
SCHEMBL6417242 0.71 HSD17B2 (0.63) MEN1KMT2AHSD17B2POLBHPGD
SCHEMBL27416257 0.71 MEN1 (0.49) TACR1MEN1KMT2AHSD17B2POLB
SCHEMBL3996160 0.70 HSD17B2 (0.61) MEN1KMT2AHSD17B2POLBHPGD
SCHEMBL27535141 0.70 MEN1 (0.48) TACR1MEN1KMT2AHSD17B2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8044067-B2 Isoquinolines as IGF-1R inhibitors ANALYTECON S.A. (CH) 2011-10-25 US disclosed
EP-1931636-B1 ISOQUINOLINES AS IGF-1R INHIBITORS ANALYTECON SA (CH) 2011-04-13 EP disclosed
US-20090099229-A1 Isoquinolines as IGF-1R Inhibitors ANALYTECON S.A (CH) 2009-04-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090099229-A1 Isoquinolines as IGF-1R Inhibitors IGF1R, IGFBP1, IGF2BP1 TACR1 1191/4885MEN1 893/4885KMT2A 1238/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.