SCHEMBL1573697

SCHEMBL1573697

Cc1cc(Cl)nc2[nH]nc(OC(=O)N3CCC(F)(F)CC3)c12

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 3/20 0.37
TSHR P16473 2/20 0.37
POLB P06746 1/20 0.36
LRRK2 Q5S007 2/20 0.32
ENPP2 Q13822 2/20 0.32
ATXN2 Q99700 2/20 0.32
LMNA P02545 1/20 0.31
APP P05067 1/20 0.31
JAK1 P23458 1/20 0.31
ACACB O00763 3/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PTGER4 P35408 1/20 0.31
PAK4 O96013 1/20 0.30
CYP3A4 P08684 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1573988 0.88 TSHR (0.33) TSHRPOLBJAK1ACACBL3MBTL1
SCHEMBL1574115 0.84 GAA (0.41) TSHRPOLBLMNACYP3A4SMN1; SMN2
SCHEMBL1573472 0.82 SPR (0.36)
SCHEMBL1573836 0.82 GAA (0.36) ACACBL3MBTL1CYP3A4SMN1; SMN2
SCHEMBL1573883 0.72 GAA (0.41) TSHRLMNACYP3A4SMN1; SMN2
SCHEMBL1573859 0.72 GAA (0.41) TSHRLMNACYP3A4SMN1; SMN2
SCHEMBL1573785 0.71 SPR (0.37)
SCHEMBL1573851 0.71 SPR (0.37)
SCHEMBL1574095 0.70 HRH3 (0.40) L3MBTL1SMN1; SMN2
SCHEMBL1573815 0.70 GAA (0.43) TSHRLMNAL3MBTL1CYP3A4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1713779-B1 INDAZOLE DERIVATIVES AS INHIBITORS OF HORMONE-SENSITIVE LIPASES SANOFI AVENTIS DEUTSCHLAND (DE) 2011-04-13 EP disclosed