Bromide

Bromide

SCHEMBL15775161

Br.Nc1nc2c(s1)CNCC2

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A known ✓ P08913 3/20 0.38
ADRA2B known ✓ P18089 2/20 0.38
ADRA2C known ✓ P18825 2/20 0.38
ADRA1A known ✓ P35348 2/20 0.38
ADRB2 known ✓ P07550 1/20 0.36
HTR1A known ✓ P08908 1/20 0.36
HTR1B known ✓ P28222 1/20 0.36
SIGMAR1 known ✓ Q99720 1/20 0.36
APOBEC3A P31941 1/20 0.50
APOBEC3G Q9HC16 1/20 0.50
DRD2 P14416 5/20 0.41
RAD52 P43351 2/20 0.40
RECQL P46063 1/20 0.40
HDAC2 Q92769 1/20 0.38
DRD3 P35462 5/20 0.38
MAPT P10636 3/20 0.38
LMNA P02545 2/20 0.38
HTR2A P28223 2/20 0.38
HRH1 P35367 2/20 0.38
OPRK1 P41145 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL14990906 1.00 APOBEC3A (0.50) APOBEC3AAPOBEC3GDRD2RAD52RECQL
SCHEMBL172067 0.98 APOBEC3A (0.52) APOBEC3AAPOBEC3GDRD2RAD52RECQL
Hydrochloric Acid SCHEMBL1202789 0.96 APOBEC3A (0.50) APOBEC3AAPOBEC3GDRD2RAD52RECQL
Hydrochloric Acid SCHEMBL15240369 0.96 APOBEC3A (0.50) APOBEC3AAPOBEC3GDRD2RAD52RECQL
Bromide SCHEMBL3309184 0.89 APOBEC3A (0.56) APOBEC3AAPOBEC3GDRD2RAD52RECQL
SCHEMBL12101179 0.87 APOBEC3A (0.58) APOBEC3AAPOBEC3GDRD2RAD52RECQL
Bromide SCHEMBL7283805 0.86 APOBEC3A (0.57) APOBEC3AAPOBEC3GDRD2RAD52RECQL
Bromide SCHEMBL14990640 0.86 APOBEC3A (0.57) APOBEC3AAPOBEC3GDRD2RAD52RECQL
SCHEMBL3307726 0.84 APOBEC3A (0.59) APOBEC3AAPOBEC3GDRD2RAD52RECQL
Trifluoroacetic Acid SCHEMBL31143352 0.83 HDAC2 (0.42) APOBEC3AAPOBEC3GDRD2RAD52RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11993595-B2 Compounds MISSION THERAPEUTICS LIMITED (GB) 2024-05-28 US disclosed
CN-111592534-B New compounds 特殊治疗有限公司 2023-06-30 CN disclosed
US-20230052191-A1 NOVEL COMPOUNDS MISSION THERAPEUTICS LTD (GB) 2023-02-16 US disclosed
US-11472798-B2 Compounds MISSION THERAPEUTICS LTD (GB) 2022-10-18 US disclosed
EP-3828179-A1 CYANOPYRROLIDINES AS DUB MODULATORS Mission Therapeutics Limited (GB) 2021-06-02 EP disclosed
US-20200369658-A1 NOVEL COMPOUNDS MISSION THERAPEUTICS LTD (GB) 2020-11-26 US disclosed
US-10774078-B2 Compounds MISSION THERAPEUTICS LTD (GB) 2020-09-15 US disclosed
CN-111592534-A Novel compounds 特殊治疗有限公司 2020-08-28 CN disclosed
EP-3197883-B1 NOVEL COMPOUNDS MISSION THERAPEUTICS LTD (GB) 2020-03-18 EP disclosed
CN-107001339-B Novel compounds 特殊治疗有限公司 2020-03-17 CN disclosed
US-20190330202-A1 NOVEL COMPOUNDS MISSION THERAPEUTICS LTD (GB) 2019-10-31 US disclosed
US-10392380-B2 Compounds MISSION THERAPEUTICS LIMITED (GB) 2019-08-27 US disclosed
US-20180162852-A1 NOVEL COMPOUNDS MISSION THERAPEUTICS LIMITED 2018-06-14 US disclosed
US-9926307-B2 Compounds MISSION THERAPEUTICS LTD (GB) 2018-03-27 US disclosed
US-20170247365-A1 NOVEL COMPOUNDS MISSION THERAPEUTICS LTD (GB) 2017-08-31 US disclosed
EP-3197883-A1 NOVEL COMPOUNDS Mission Therapeutics Limited (GB) 2017-08-02 EP disclosed
WO-2016046530-A1 NOVEL COMPOUNDS MISSION THERAPEUTICS LTD (GB) 2016-03-31 WO disclosed
WO-2014086478-A1 INHIBITORS OF MALT1 PROTEASE Helmholtz Zentrum München - Deutsches Forschungszentrum für Gesundheit und Umwelt (GmbH) (DE) 2014-06-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10774078-B2 Compounds UCHL1, UCHL3, UCHL5 ADRA2A 4577/4885ADRA2B 4525/4885ADRA2C 4434/4885
US-11472798-B2 Compounds UCHL1, UCHL3, UCHL5 ADRA2A 4577/4885ADRA2B 4525/4885ADRA2C 4434/4885
US-20180162852-A1 NOVEL COMPOUNDS UCHL1, UCHL3, UCHL5 ADRA2A 4357/4885ADRA2B 4266/4885ADRA2C 4205/4885
US-10392380-B2 Compounds UCHL1, UCHL3, UCHL5 ADRA2A 4577/4885ADRA2B 4525/4885ADRA2C 4434/4885
US-11993595-B2 Compounds UCHL1, UCHL3, UCHL5 ADRA2A 4577/4885ADRA2B 4525/4885ADRA2C 4434/4885
US-20200369658-A1 NOVEL COMPOUNDS UCHL1, UCHL3, UCHL5 ADRA2A 4357/4885ADRA2B 4266/4885ADRA2C 4205/4885
US-20190330202-A1 NOVEL COMPOUNDS UCHL1, UCHL3, UCHL5 ADRA2A 4357/4885ADRA2B 4266/4885ADRA2C 4205/4885
US-20170247365-A1 NOVEL COMPOUNDS UCHL1, UCHL3, UCHL5 ADRA2A 4357/4885ADRA2B 4266/4885ADRA2C 4205/4885
US-20230052191-A1 NOVEL COMPOUNDS UCHL1, UCHL3, UCHL5 ADRA2A 4357/4885ADRA2B 4266/4885ADRA2C 4205/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.