SCHEMBL15775256

SCHEMBL15775256

Cc1ccc(-c2nc(=O)c3cnccc3[nH]2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.49
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
PARP1 P09874 4/20 0.44
TNKS O95271 3/20 0.44
TNKS2 Q9H2K2 3/20 0.44
MAPK13 O15264 1/20 0.44
GCGR P47871 1/20 0.44
MAPK12 P53778 1/20 0.44
MAPK11 Q15759 1/20 0.44
MAPK14 Q16539 1/20 0.44
KDM4E B2RXH2 2/20 0.43
KMT2A Q03164 2/20 0.43
AURKA O14965 1/20 0.43
ALDH1A1 P00352 3/20 0.42
PKM P14618 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
HPGD P15428 1/20 0.42
MAPT P10636 2/20 0.40
KDM4C Q9H3R0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15775358 0.88 AURKA (0.46) NPC1RAB9APARP1TNKSTNKS2
SCHEMBL15775257 0.85 ALDH1A1 (0.60) NPC1RAB9APARP1TNKSTNKS2
SCHEMBL15775281 0.85 KDM4C (0.56) ACHENPC1RAB9APARP1TNKS
SCHEMBL15775687 0.80 TNKS (0.59) NPC1RAB9APARP1TNKSTNKS2
Hydrochloric Acid SCHEMBL7280780 0.77 NPC1 (0.56) NPC1RAB9APARP1TNKSTNKS2
SCHEMBL15775258 0.77 TNKS (0.67) NPC1RAB9APARP1TNKSTNKS2
SCHEMBL11306011 0.75 MEN1 (0.49) NPC1RAB9APARP1TNKSTNKS2
SCHEMBL16331618 0.75 ALDH1A1 (0.71) NPC1RAB9AKDM4EKMT2AAURKA
SCHEMBL15775972 0.73 TNKS (0.51) NPC1RAB9APARP1TNKSTNKS2
SCHEMBL15775362 0.73 KDM4C (0.74) RAB9APARP1TNKSTNKS2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO disclosed