SCHEMBL15775360

SCHEMBL15775360

COc1cccc(C(N)C#N)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 3/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
TAAR1 Q96RJ0 2/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP3A4 P08684 1/20 0.46
PARP1 P09874 1/20 0.43
PRSS1 P07477 1/20 0.43
PRSS2 P07478 1/20 0.43
PRSS3 P35030 1/20 0.43
ACHE P22303 1/20 0.42
CASR P41180 2/20 0.42
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
KMT2A Q03164 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5740866 0.98 AOC3 (0.46) AOC3L3MBTL1TAAR1ALDH1A1CYP3A4
Hydrochloric Acid SCHEMBL5740863 0.98 AOC3 (0.46) AOC3L3MBTL1TAAR1ALDH1A1CYP3A4
SCHEMBL11565961 0.82 L3MBTL1 (0.50) AOC3L3MBTL1TAAR1ALDH1A1CYP3A4
SCHEMBL17466002 0.81 ALDH1A1 (0.48) AOC3L3MBTL1ALDH1A1CYP3A4PARP1
SCHEMBL5384948 0.81 ALOX5 (0.49) ALDH1A1KMT2A
SCHEMBL2178067 0.80 AOC3 (0.43) AOC3L3MBTL1TAAR1ALDH1A1CASR
SCHEMBL954319 0.80 CASR (0.46) AOC3L3MBTL1TAAR1ALDH1A1CYP3A4
SCHEMBL7652207 0.79 KMT2A (0.49) AOC3L3MBTL1TAAR1ACHECASR
Hydrochloric Acid SCHEMBL5744406 0.79 ALOX5 (0.48) ALDH1A1KMT2A
SCHEMBL29061992 0.79 KMT2A (0.49) AOC3L3MBTL1TAAR1ACHECASR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150299143-A1 SUBSTITUTED TRIAZOLE AND IMIDAZOLE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2015-10-22 US claimed
EP-2925746-A1 SUBSTITUTED TRIAZOLE AND IMIDAZOLE COMPOUNDS F. Hoffmann-La Roche AG (CH) 2015-10-07 EP claimed
WO-2014086663-A1 SUBSTITUTED TRIAZOLE AND IMIDAZOLE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2014-06-12 WO claimed
US-20150299143-A1 SUBSTITUTED TRIAZOLE AND IMIDAZOLE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2015-10-22 US disclosed
EP-2925746-A1 SUBSTITUTED TRIAZOLE AND IMIDAZOLE COMPOUNDS F. Hoffmann-La Roche AG (CH) 2015-10-07 EP disclosed
WO-2014086663-A1 SUBSTITUTED TRIAZOLE AND IMIDAZOLE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2014-06-12 WO disclosed
CN-1324006-C Beta-amino acid nitrile derivs. HOFFMANN LA ROCHE (CH) 2007-07-04 CN disclosed
CN-1436168-A Beta-amino acid nitrile derivs. HOFFMANN LA ROCHE (CH) 2003-08-13 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150299143-A1 SUBSTITUTED TRIAZOLE AND IMIDAZOLE COMPOUNDS HDAC7, PSMB7, IKZF3 AOC3 2479/4885L3MBTL1 3540/4885TAAR1 1677/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.