SCHEMBL15775552

SCHEMBL15775552

O=C1CN(c2ccccc2)Cc2cnccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.42
PDE3B Q13370 2/20 0.41
PDE3A Q14432 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
MAPT P10636 2/20 0.41
EED O75530 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
HTT P42858 2/20 0.38
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
TIPARP Q7Z3E1 2/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15775155 0.88 CYP11B2 (0.46) CYP11B2PDE3BPDE3ANPC1RAB9A
SCHEMBL15777255 0.85 CA12 (0.42) CYP11B2PDE3BPDE3AMAPTCA12
SCHEMBL15775371 0.81 TIPARP (0.43) PDE3BPDE3ACA12CA2CA9
SCHEMBL4987770 0.73 MITF (0.40) PDE3BPDE3ARAB9AMAPTMAOA
SCHEMBL10311113 0.72 EED (0.41) CYP11B2PDE3BPDE3ANPC1RAB9A
SCHEMBL15776946 0.70 TIPARP (0.43) CA12CA2CA9CYP2C9TIPARP
SCHEMBL6591115 0.68 EED (0.75) NPC1RAB9AMAPTEEDALDH1A1
SCHEMBL8866710 0.68 CYP11B2 (0.56) CYP11B2NPC1RAB9AMAOAMAOB
SCHEMBL2185054 0.67 MEN1 (0.67) NPC1RAB9AMAPTEEDALDH1A1
SCHEMBL30466979 0.67 MEN1 (0.67) NPC1RAB9AMAPTEEDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO disclosed