SCHEMBL15775371

SCHEMBL15775371

O=C1CN(c2ccc(C(F)(F)F)cc2)Cc2cnccc21

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TIPARP Q7Z3E1 1/20 0.43
CYP3A4 P08684 7/20 0.40
GRM2 Q14416 2/20 0.39
PDE2A O00408 1/20 0.38
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
KIF11 P52732 1/20 0.37
CACNA1B Q00975 2/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HIF1A Q16665 2/20 0.36
TSHR P16473 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CA12 O43570 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15776946 0.89 TIPARP (0.43) TIPARPCYP3A4GRM2PDE2AKIF11
SCHEMBL15777255 0.82 CA12 (0.42) TIPARPPDE3BPDE3ACA12CA2
SCHEMBL15775552 0.81 CYP11B2 (0.42) TIPARPCYP3A4PDE3BPDE3ATSHR
SCHEMBL30822812 0.70 CA12 (0.49) CYP3A4CA12CA2CA9
SCHEMBL15775155 0.70 CYP11B2 (0.46) TIPARPCYP3A4PDE3BPDE3ATSHR
SCHEMBL4987770 0.68 MITF (0.40) TIPARPCYP3A4PDE3BPDE3A
SCHEMBL4323285 0.65 CYP1A2 (0.53) PDE3BPDE3ACYP1A2
SCHEMBL29792666 0.65 CYP1A2 (0.53) PDE3BPDE3ACYP1A2
SCHEMBL30947594 0.63 CYP11B2 (0.41) TIPARPPDE3BPDE3AHDAC1HDAC2
SCHEMBL28650484 0.62 CA12 (0.65) CYP3A4GRM2CA12CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO disclosed