SCHEMBL1583554

SCHEMBL1583554

CC1(F)CNC(=O)NC1=O

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.32
LMNA P02545 1/20 0.31
CRBN Q96SW2 1/20 0.31
MMP2 P08253 1/20 0.30
MMP9 P14780 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25417178 0.85
SCHEMBL6221243 0.75 SMN1; SMN2 (0.34) SMN1; SMN2LMNACRBNMMP2MMP9
SCHEMBL11375741 0.75 CRBN (0.33) CRBN
SCHEMBL48327 0.71 LMNA (0.36) SMN1; SMN2LMNACRBNMMP2MMP9
SCHEMBL28864845 0.71 SMN1; SMN2 (0.32) SMN1; SMN2LMNACRBNMMP2MMP9
SCHEMBL29110862 0.71 CRBN (0.31) CRBN
SCHEMBL2473210 0.71 SMN1; SMN2 (0.32) SMN1; SMN2LMNACRBNMMP2MMP9
SCHEMBL29110865 0.71 CRBN (0.31) CRBN
SCHEMBL24227250 0.70 SMN1; SMN2 (0.31) SMN1; SMN2LMNACRBN
SCHEMBL4339901 0.68 SMN1; SMN2 (0.30) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1374911-B1 AGENTS FOR MEASURING PYRIMIDINE METABOLIZABILITY OTSUKA PHARMA CO LTD (JP) 2013-10-16 EP claimed
EP-2512491-B1 HBV ANTISENSE INHIBITORS GLAXO GROUP LTD (GB) 2017-10-11 EP disclosed
US-8883121-B2 Oral preparation useful in measurement capacity to metabolize pyridine OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2014-11-11 US disclosed
US-8598334-B2 HBV antisense inhibitors GLAXO GROUP LIMITED (GB) 2013-12-03 US disclosed
EP-2512491-A1 HBV ANTISENSE INHIBITORS Glaxo Group Limited (GB) 2012-10-24 EP disclosed
US-20120207709-A1 HBV ANTISENSE INHIBITORS GLAXO GROUP LIMITED (GB) 2012-08-16 US disclosed
EP-1920786-B1 ORAL PREPARATION FOR MEASURING PYRIMIDINE METABOLIC CAPACITY OTSUKA PHARMA CO LTD (JP) 2011-10-05 EP disclosed
WO-2011047312-A1 HBV ANTISENSE INHIBITORS GLAXO GROUP LIMITED (GB) 2011-04-21 WO disclosed
US-20080233048-A1 Powder by mixing and pulverizing an isotope-labeled uracil, or metabolite labeled with an isotope of carbon atoms, oxygen atoms, or nitrogen atoms and mannitol; time required for the determination and number of measurements can be reduced, decreasing the burden on patients OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-09-25 US disclosed
EP-1920786-A1 ORAL PREPARATION USEFUL IN MEASURING CAPACITY TO METABOLIZE PYRIDINE Otsuka Pharmaceutical Co., Ltd. (JP) 2008-05-14 EP disclosed
US-20030068272-A1 Preparation for determining pyrimidine metabolic capacity OTSUKA PHARMACEUTICAL CO., LTD. 2003-04-10 US disclosed
US-4246411-A ANTICARCINOGENIC AGENTS PCR INCORPORATED (US) 1981-01-20 US disclosed
US-4029661-A OR ALCOHOL SOLVENTSFLUORINATION PCR, INC. (US) 1977-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120207709-A1 HBV ANTISENSE INHIBITORS HAVCR2, BCDIN3D, HLA-B SMN1; SMN2 2335/4885LMNA 1497/4885CRBN 4470/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.