SCHEMBL1583909

SCHEMBL1583909

CC(C)COC(=O)N1CCN(c2cccs2)C(=O)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
PKM P14618 1/20 0.40
BRD4 O60885 1/20 0.38
ADORA2B P29275 1/20 0.38
KIT P10721 1/20 0.38
HPGD P15428 3/20 0.37
ALDH1A1 P00352 3/20 0.37
HTT P42858 2/20 0.37
KDM4E B2RXH2 2/20 0.37
LMNA P02545 2/20 0.37
ALOX12 P18054 2/20 0.37
CASP1 P29466 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 2/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
TDP1 Q9NUW8 2/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1583906 0.80 GPR119 (0.43) ALDH1A1KDM4ELMNAPOLBMEN1
SCHEMBL1583651 0.79 CYP1A2 (0.41) ADORA2BKITHPGDALDH1A1HTT
SCHEMBL1583153 0.79 ROCK2 (0.50) KITHPGDALDH1A1KDM4ELMNA
SCHEMBL3653187 0.78 P2RX7 (0.52) SMN1; SMN2ALDH1A1LMNATSHRP2RX4
SCHEMBL1583384 0.77 KDM4E (0.48) KITHPGDALDH1A1KDM4ELMNA
SCHEMBL1663016 0.77 P2RX7 (0.53) HSD17B10KITALDH1A1TSHRP2RX4
SCHEMBL1583489 0.77 SCN9A (0.51) SMN1; SMN2ALDH1A1KDM4ELMNATSHR
SCHEMBL1583535 0.76 HRH3 (0.49) CYP3A4HDAC2
SCHEMBL1583833 0.76 TSHR (0.37) HSD17B10KITHPGDALDH1A1HTT
SCHEMBL1583149 0.76 DPP4 (0.49) HSD17B10ALDH1A1KDM4ENPSR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011041713-A2 PIPERAZINYL ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2011-04-07 WO disclosed