SCHEMBL15890232

SCHEMBL15890232

Cc1noc(C)c1NC(=O)Oc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.53
IDO1 P14902 1/20 0.51
ALDH1A1 P00352 7/20 0.48
MAPT P10636 4/20 0.48
LPAR1 Q92633 1/20 0.47
LPAR3 Q9UBY5 1/20 0.47
RAD51 Q06609 1/20 0.47
RIPK1 Q13546 1/20 0.46
BRD2 P25440 1/20 0.45
KDM4E B2RXH2 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
THRB P10828 1/20 0.44
GFER P55789 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
GAA P10253 2/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
RAB9A P51151 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1011568 0.79 IDO1 (0.54) IDO1ALDH1A1MAPTRAD51KDM4E
SCHEMBL19563752 0.79 IDO1 (0.60) IDO1ALDH1A1MAPTRAD51KDM4E
SCHEMBL8809532 0.75 PKM (0.48) IDO1ALDH1A1MAPTRAD51KDM4E
SCHEMBL897183 0.75 RAB9A (0.61) ALDH1A1KDM4EMEN1KMT2AGAA
SCHEMBL10526068 0.74 ALDH1A1 (0.56) ALDH1A1MAPTRAD51KDM4EMEN1
Hydrochloric Acid SCHEMBL8808042 0.74 PKM (0.47) IDO1ALDH1A1MAPTRAD51KDM4E
SCHEMBL2322209 0.74 ALDH1A1 (0.67) IDO1ALDH1A1MAPTKDM4EMEN1
SCHEMBL1895964 0.73 ALDH1A1 (0.53) IDO1ALDH1A1MAPTRAD51KDM4E
Hydrochloric Acid SCHEMBL1375757 0.73 BRD4 (0.45) BRD4ALDH1A1MAPTRIPK1BRD2
SCHEMBL17736670 0.72 IDO1 (0.59) IDO1ALDH1A1MAPTRAD51KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014111871-A1 4,5-DIHYDROISOXAZOLE DERIVATIVES AS NAMPT INHIBITORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2014-07-24 WO disclosed