SCHEMBL15919180

SCHEMBL15919180

CC(C)(C)OC(=O)NCCCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCOCCOCCOCCOCCC(=O)O

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.49
CTSK P43235 4/20 0.49
SIRT5 Q9NXA8 1/20 0.48
GLP1R P43220 8/20 0.47
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
MEN1 O00255 1/20 0.46
GAA P10253 1/20 0.46
KMT2A Q03164 1/20 0.46
CAPN1 P07384 1/20 0.46
TDP1 Q9NUW8 1/20 0.42
CXCR3 P49682 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23077723 1.00 CTSS (0.49) CTSSCTSKSIRT5GLP1RCA1
SCHEMBL26689262 0.94 GLP1R (0.52) CTSSCTSKSIRT5GLP1RCA1
SCHEMBL26689380 0.94 GLP1R (0.52) CTSSCTSKSIRT5GLP1RCA1
SCHEMBL26689259 0.94 GLP1R (0.52) CTSSCTSKSIRT5GLP1RCA1
SCHEMBL26689385 0.94 GLP1R (0.52) CTSSCTSKSIRT5GLP1RCA1
SCHEMBL19543629 0.92 CTSS (0.53) CTSSCTSKSIRT5CA1CA2
SCHEMBL24667758 0.92 GLP1R (0.55) CTSSCTSKSIRT5GLP1RCA1
SCHEMBL26689110 0.89 GLP1R (0.49) CTSSCTSKSIRT5GLP1RCA1
SCHEMBL26689108 0.89 GLP1R (0.49) CTSSCTSKSIRT5GLP1RCA1
SCHEMBL26689250 0.89 GLP1R (0.49) CTSSCTSKSIRT5GLP1RCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10947289-B2 Glyco-modified atrial natriuretic peptide DAIICHI SANKYO COMPANY, LIMITED (JP) 2021-03-16 US disclosed
US-10947289-B2 Glyco-modified atrial natriuretic peptide DAIICHI SANKYO COMPANY, LIMITED (JP) 2021-03-16 US disclosed
US-20210040170-A1 GLYCO-MODIFIED ATRIAL NATRIURETIC PEPTIDE DAIICHI SANKYO COMPANY, LIMITED (JP) 2021-02-11 US disclosed
US-20210040170-A1 GLYCO-MODIFIED ATRIAL NATRIURETIC PEPTIDE DAIICHI SANKYO COMPANY, LIMITED (JP) 2021-02-11 US disclosed
EP-2949665-B1 GLYCOSYLATION ATRIAL NATRIURETIC PEPTIDE DAIICHI SANKYO CO LTD (JP) 2018-02-28 EP disclosed
EP-2949665-B1 GLYCOSYLATION ATRIAL NATRIURETIC PEPTIDE DAIICHI SANKYO CO LTD (JP) 2018-02-28 EP disclosed
US-20160017015-A1 GLYCO-MODIFIED ATRIAL NATRIURETIC PEPTIDE DAIICHI SANKYO COMPANY, LIMITED (JP) 2016-01-21 US disclosed
US-20160017015-A1 GLYCO-MODIFIED ATRIAL NATRIURETIC PEPTIDE DAIICHI SANKYO COMPANY, LIMITED (JP) 2016-01-21 US disclosed
EP-2949665-A1 GLYCOSYLATION ATRIAL NATRIURETIC PEPTIDE DAIICHI SANKYO COMPANY, LIMITED (JP) 2015-12-02 EP disclosed
EP-2949665-A1 GLYCOSYLATION ATRIAL NATRIURETIC PEPTIDE DAIICHI SANKYO COMPANY, LIMITED (JP) 2015-12-02 EP disclosed
WO-2014115797-A1 GLYCOSYLATION ATRIAL NATRIURETIC PEPTIDE 第一三共株式会社 (JP) 2014-07-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10947289-B2 Glyco-modified atrial natriuretic peptide NPPA, NPR1, NPR3 CTSS 3994/4885CTSK 3394/4885SIRT5 1560/4885
US-20210040170-A1 GLYCO-MODIFIED ATRIAL NATRIURETIC PEPTIDE NPPA, NPR1, NPR3 CTSS 3994/4885CTSK 3394/4885SIRT5 1560/4885
US-20160017015-A1 GLYCO-MODIFIED ATRIAL NATRIURETIC PEPTIDE NPPA, NPR1, NPR3 CTSS 3994/4885CTSK 3394/4885SIRT5 1560/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.