SCHEMBL15922883

SCHEMBL15922883

CC(C)(C)N1CCN(c2ccc(N)c(N)c2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 9/20 0.49
GAA P10253 5/20 0.49
MAPK1 P28482 3/20 0.49
HTT P42858 3/20 0.49
KDM4E B2RXH2 3/20 0.49
PTK2B Q14289 2/20 0.49
RECQL P46063 2/20 0.49
RAD52 P43351 2/20 0.45
LMNA P02545 5/20 0.43
ALDH1A1 P00352 4/20 0.43
S100B P04271 2/20 0.43
KMT2A Q03164 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
MEN1 O00255 1/20 0.43
PKM P14618 1/20 0.43
ALOX15 P16050 1/20 0.43
LGMN Q99538 3/20 0.42
SIRT6 Q8N6T7 1/20 0.42
ADRA2C P18825 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11291219 0.82 ALDH1A1 (0.43) MAPTGAAMAPK1HTTKDM4E
SCHEMBL1476346 0.79 MAPT (0.62) MAPTGAAMAPK1HTTKDM4E
SCHEMBL29745032 0.79 GAA (0.73) MAPTGAAMAPK1HTTKDM4E
SCHEMBL76547 0.79 GAA (0.73) MAPTGAAMAPK1HTTKDM4E
SCHEMBL3986308 0.79 MAPT (0.72) MAPTMAPK1RECQLLMNAALDH1A1
SCHEMBL16654817 0.79 MAPT (0.57) MAPTRECQLLMNAALDH1A1KMT2A
SCHEMBL30822482 0.79 ADRA2C (0.66) MAPTGAAMAPK1HTTKDM4E
Ammonia Solution, Strong SCHEMBL14746306 0.78 GAA (0.71) MAPTGAAMAPK1HTTKDM4E
SCHEMBL24625570 0.78 GAA (0.39) MAPTGAAMAPK1HTTKDM4E
SCHEMBL7372826 0.77 MAPT (0.68) MAPTGAAMAPK1HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016183150-A1 NOVEL SIGMA-2 RECEPTOR BINDERS AND THEIR METHOD OF USE TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2016-11-17 WO disclosed
EP-2951153-A1 SELECTIVE HDAC3 INHIBITORS Acetylon Pharmaceuticals, Inc. (US) 2015-12-09 EP disclosed
WO-2014121062-A1 SELECTIVE HDAC3 INHIBITORS ACETYLON PHARMACEUTICALS, INC. (US) 2014-08-07 WO disclosed