SCHEMBL15927802

SCHEMBL15927802

N[C@@H](Cc1ccccc1)C(=O)N1CCC2CCCC2C1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 5/20 0.58
HDAC8 Q9BY41 3/20 0.56
DPP8 Q6V1X1 2/20 0.53
DPP9 Q86TI2 2/20 0.53
DPP7 Q9UHL4 2/20 0.53
FAP Q12884 1/20 0.53
OPRD1 P41143 1/20 0.53
POLB P06746 1/20 0.52
TACR1 P25103 1/20 0.48
ROCK2 O75116 1/20 0.48
CYP3A4 P08684 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21408995 0.85 DPP7 (0.49) DPP4DPP7
SCHEMBL5891540 0.83 HDAC8 (0.60) DPP4HDAC8DPP8DPP9DPP7
SCHEMBL6052747 0.83 HDAC8 (0.59) DPP4HDAC8DPP8DPP9DPP7
SCHEMBL4095232 0.83 HDAC8 (0.59) DPP4HDAC8DPP8DPP9DPP7
SCHEMBL4086820 0.83 HDAC8 (0.59) DPP4HDAC8DPP8DPP9DPP7
Hydrochloric Acid SCHEMBL5891327 0.82 HDAC8 (0.61) DPP4HDAC8DPP8DPP9DPP7
SCHEMBL6161830 0.80 OPRD1 (0.65) DPP4HDAC8DPP8DPP9DPP7
SCHEMBL3133533 0.80 OPRD1 (0.65) DPP4HDAC8DPP8DPP9DPP7
SCHEMBL21431185 0.80 HPGD (0.69) DPP4HDAC8DPP8DPP9DPP7
SCHEMBL6705226 0.80 HDAC8 (0.56) DPP4HDAC8DPP8DPP9DPP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9062057-B2 CCR5 antagonists for treating HIV PURDUE RESEARCH FOUNDATION (US) 2015-06-23 US disclosed
US-20140221420-A1 CCR5 ANTAGONISTS FOR TREATING HIV PURDUE RESEARCH FOUNDATION (US) 2014-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140221420-A1 CCR5 ANTAGONISTS FOR TREATING HIV CCR5, CXCR4, CXCR3 DPP4 1694/4885HDAC8 1402/4885DPP8 732/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.