SCHEMBL15929129

SCHEMBL15929129

CCc1ccc(C(=O)Oc2ccc3cc([C@H](C)C(=O)Oc4ccc(C(N)=S)cc4)ccc3c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.45
AKR1C2 P52895 2/20 0.45
PTGS2 P35354 5/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
PRSS1 P07477 1/20 0.41
ACR P10323 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HGFAC Q04756 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19341478 0.90 AKR1C3 (0.46) AKR1C3AKR1C2PTGS2TDP1L3MBTL1
SCHEMBL19341483 0.88 AKR1C3 (0.48) AKR1C3AKR1C2PTGS2TDP1L3MBTL1
SCHEMBL15929140 0.85 PTGS2 (0.38) AKR1C3AKR1C2PTGS2PRSS1ACR
SCHEMBL15929023 0.85 AKR1C3 (0.43) AKR1C3AKR1C2PTGS2PRSS1ACR
Atb-346 SCHEMBL23643163 0.83 PTGS2 (0.63) AKR1C3AKR1C2PTGS2TDP1L3MBTL1
Atb-346 SCHEMBL29358559 0.83 PTGS2 (0.63) AKR1C3AKR1C2PTGS2TDP1L3MBTL1
Atb-346 SCHEMBL2883303 0.83 PTGS2 (0.63) AKR1C3AKR1C2PTGS2TDP1L3MBTL1
Atb-346 SCHEMBL31566275 0.83 PTGS2 (0.63) AKR1C3AKR1C2PTGS2TDP1L3MBTL1
Atb-346 SCHEMBL29596141 0.83 PTGS2 (0.63) AKR1C3AKR1C2PTGS2TDP1L3MBTL1
SCHEMBL15929139 0.82 PTGS2 (0.44) AKR1C3AKR1C2PTGS2TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170260124-A1 NO- AND H2S- RELEASING COMPOUNDS RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK 2017-09-14 US disclosed
US-9688607-B2 No- and H2S-releasing compounds RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK (US) 2017-06-27 US disclosed
US-20140221316-A1 NO- AND H2S- RELEASING COMPOUNDS RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK (US) 2014-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140221316-A1 NO- AND H2S- RELEASING COMPOUNDS PTGS1, NOS2, NOS1 AKR1C3 2456/4885AKR1C2 2270/4885PTGS2 4/4885
US-20170260124-A1 NO- AND H2S- RELEASING COMPOUNDS NOS2, NOS3, NOS1 AKR1C3 2812/4885AKR1C2 2722/4885PTGS2 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.