SCHEMBL15933682

SCHEMBL15933682

CC(C)(C)OC(=O)N1CCn2cc(-c3cccnc3)nc2C1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.52
GPR119 Q8TDV5 2/20 0.48
KIT P10721 1/20 0.47
P2RX7 Q99572 2/20 0.44
GRM5 P41594 1/20 0.44
GRM1 Q13255 1/20 0.44
CKS1B P61024 2/20 0.43
SKP1 P63208 2/20 0.43
SKP2 Q13309 2/20 0.43
POLB P06746 1/20 0.42
WDR5 P61964 1/20 0.41
CCNA2 P20248 1/20 0.41
CDK2 P24941 1/20 0.41
KDM1A O60341 1/20 0.41
NAMPT P43490 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP3A5 P20815 1/20 0.41
MAPK1 P28482 1/20 0.41
NR1H2 P55055 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15933469 0.88 GPR119 (0.43) GBA1GPR119KITP2RX7CKS1B
SCHEMBL4399124 0.88 GPR119 (0.46) GPR119P2RX7GRM1POLBMAPK1
SCHEMBL17298980 0.82 F2RL1 (0.45) P2RX7GRM5GRM1KDM1ANAMPT
SCHEMBL15933636 0.81 P2RX7 (0.43) GPR119P2RX7CKS1BSKP1SKP2
SCHEMBL2813207 0.80 SMARCA2 (0.53) GPR119P2RX7CKS1BSKP1SKP2
SCHEMBL15933695 0.80 EGLN2 (0.48) GPR119P2RX7
SCHEMBL15933586 0.79 GPR119 (0.52) GPR119NR1H2
SCHEMBL23390025 0.79 GRM5 (0.44) GPR119P2RX7GRM5CKS1BSKP1
SCHEMBL29796413 0.79 GRM5 (0.44) GPR119P2RX7GRM5CKS1BSKP1
SCHEMBL4399119 0.76 NR1H2 (0.55) GBA1GPR119KITGRM5GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014117318-A1 NOVEL TRIAZOLE ANTIFUNGAL COMPOUNDS, AND PHARMACEUTICAL COMPOSITION, PREPARATION METHOD, AND APPLICATION THEREOF 中国科学院上海药物研究所 (CN) 2014-08-07 WO disclosed