SCHEMBL15935550

SCHEMBL15935550

CC(C)(C)c1ccc2c(c1)CC1(C2)OC(=O)Cc2nccnc21

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 10/20 0.33
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
ADRA1D P25100 1/20 0.31
HTR1D P28221 1/20 0.31
HTR1B P28222 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15935556 0.85 AVPR1A (0.40) AVPR1A
SCHEMBL15935552 0.79 DGAT1 (0.30) AVPR1A
SCHEMBL13015186 0.79 ADRA2A (0.33) AVPR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL13015187 0.70 CALCRL (0.38)
SCHEMBL13015171 0.69 GRIN2D (0.32)
SCHEMBL13015184 0.68 KCNH2 (0.39) AVPR1A
SCHEMBL13015185 0.65 DGAT1 (0.30) AVPR1A
SCHEMBL15935551 0.65 CALCRL (0.36)
SCHEMBL26042425 0.63 ALDH1A1 (0.33)
SCHEMBL15935915 0.63 AVPR1A (0.38) AVPR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8796260-B2 Imidazobenzazepine CGRP receptor antagonists MERCK SHARP & DOHME CORP. (US) 2014-08-05 US disclosed