Guanine

Guanine

SCHEMBL15948930

Nc1nc2[nH]cnc2c(=O)[nH]1.O=P(O)(O)S

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
LMNA P02545 1/20 0.50
GLA P06280 1/20 0.50
PMP22 Q01453 1/20 0.50
HSD17B10 Q99714 1/20 0.50
PNP P00491 6/20 0.44
HPRT1 P00492 8/20 0.41
DYRK1A Q13627 1/20 0.41
AKR1B1 P15121 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Guanine SCHEMBL663745 0.94 KDM4E (0.53) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL76053 0.94 KDM4E (0.53) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL5372452 0.92 KDM4E (0.51) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL4658042 0.89 ALDH1A1 (0.61) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL5259 0.89 ALDH1A1 (0.61) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL101892 0.88 KDM4E (0.48) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL27542045 0.87 HSD17B10 (0.56) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL865492 0.87 ALDH1A1 (0.59) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL2895087 0.87 ALDH1A1 (0.59) KDM4EALDH1A1LMNAGLAPMP22
Guanine SCHEMBL21611717 0.87 ALDH1A1 (0.59) KDM4EALDH1A1LMNAGLAPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2380897-B1 RNAi modulation of ApoB and uses thereof ALNYLAM PHARMACEUTICALS INC (US) 2015-05-13 EP disclosed
EP-2377873-B1 RNAi modulation of ApoB and uses thereof ALNYLAM PHARMACEUTICALS INC (US) 2014-08-20 EP disclosed
CN-101133074-A RNAi modulation of APOB and uses thereof ALNYLAM PHARMACEUTICALS INC (US) 2008-02-27 CN disclosed