SCHEMBL15958673

SCHEMBL15958673

Cc1cccc(C(C)Cc2cccnc2)c1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.44
ADRA2A P08913 4/20 0.43
ADRA2B P18089 4/20 0.43
ADRA2C P18825 4/20 0.43
ADRA1A P35348 3/20 0.43
ADRA1B P35368 3/20 0.43
ADRA1D P25100 2/20 0.43
TSHR P16473 2/20 0.43
KCNH2 Q12809 1/20 0.43
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTT P42858 2/20 0.42
SLC6A2 P23975 1/20 0.42
HTR7 P34969 1/20 0.42
FDPS P14324 1/20 0.42
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1157247 0.85 GAA (0.48) P2RX7ADRA2AADRA2BADRA2CADRA1A
SCHEMBL12637595 0.84 P2RX7 (0.43) P2RX7ADRA2AADRA2BADRA2CADRA1A
SCHEMBL6546728 0.80 SIGMAR1 (0.48) CYP2D6SLC6A2
SCHEMBL13732891 0.77 P2RX7 (0.41) P2RX7ADRA2AADRA2BADRA2CADRA1A
SCHEMBL32673069 0.74 ADRA2A (0.38) P2RX7ADRA2AADRA2BADRA2CADRA1A
SCHEMBL32673000 0.74 ADRA2A (0.38) P2RX7ADRA2AADRA2BADRA2CADRA1A
SCHEMBL12894954 0.73 SLC6A2 (0.57) CYP1A2CYP2D6SLC6A2FDPSCHRNB2
SCHEMBL290633 0.73 SLC6A2 (0.57) CYP1A2CYP2D6SLC6A2FDPSCHRNB2
SCHEMBL29669201 0.73 SLC6A2 (0.57) CYP1A2CYP2D6SLC6A2FDPSCHRNB2
SCHEMBL31570740 0.73 GAA (0.55) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8809379-B2 Selective subtype alpha 2 adrenergic agents and methods for use thereof ALLERGAN, INC. (US) 2014-08-19 US disclosed