SCHEMBL15958962

SCHEMBL15958962

Cn1cc(-c2ccc(F)cc2)c2ccc(C=O)cc21

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.53
TDO2 P48775 1/20 0.53
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 2/20 0.46
PARG Q86W56 1/20 0.42
CYP2A6 P11509 2/20 0.42
PTGS1 P23219 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SCN9A Q15858 9/20 0.40
SCN5A Q14524 4/20 0.40
PGR P06401 1/20 0.40
PRKCA P17252 1/20 0.39
GSK3B P49841 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22159339 0.85 SCN9A (0.51) IDO1TDO2KDM4EALDH1A1CYP2A6
SCHEMBL31632863 0.85 IDO1 (0.44) IDO1TDO2KDM4EALDH1A1CYP2A6
SCHEMBL31632773 0.79 SCN9A (0.44) IDO1TDO2KDM4EALDH1A1CYP2A6
SCHEMBL121650 0.76 IDO1 (0.58) IDO1TDO2SCN9ASCN5A
SCHEMBL121418 0.76 IDO1 (0.58) IDO1TDO2KDM4EALDH1A1PTGS1
SCHEMBL16452865 0.75 ALDH1A1 (0.38) IDO1TDO2KDM4EALDH1A1MEN1
SCHEMBL19831270 0.73 CYP2A6 (0.50) KDM4EALDH1A1CYP2A6MEN1KMT2A
SCHEMBL9300549 0.73 IMPDH2 (0.57) IDO1TDO2KDM4EALDH1A1MEN1
SCHEMBL16474119 0.73 IDO1 (0.55) IDO1TDO2SCN9ASCN5A
SCHEMBL147558 0.73 IDO1 (0.58) IDO1TDO2PTGS1SCN9ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421825-B9 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2014-08-20 EP disclosed