SCHEMBL1596779

SCHEMBL1596779

CCOC(=O)C(O)Cc1ccc(OCc2ccccc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.65
LMNA P02545 1/20 0.65
PPARA Q07869 4/20 0.60
PPARG P37231 3/20 0.60
LTA4H P09960 2/20 0.60
PPARD Q03181 1/20 0.60
LAP3 P28838 1/20 0.59
ALOX5 P09917 3/20 0.57
NR1H4 Q96RI1 1/20 0.55
ALDH1A1 P00352 1/20 0.55
FFAR1 O14842 1/20 0.55
FFAR4 Q5NUL3 1/20 0.55
MAOB P27338 3/20 0.54
NR4A1 P22736 1/20 0.51
NR4A2 P43354 1/20 0.51
NR4A3 Q92570 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4756342 1.00 L3MBTL1 (0.65) L3MBTL1LMNAPPARAPPARGLTA4H
SCHEMBL5375675 1.00 L3MBTL1 (0.65) L3MBTL1LMNAPPARAPPARGLTA4H
SCHEMBL27854776 0.90 LTA4H (0.71) LMNAPPARAPPARGLTA4HPPARD
SCHEMBL6738407 0.89 LTA4H (0.57) L3MBTL1LMNAPPARAPPARGLTA4H
SCHEMBL6738411 0.89 LTA4H (0.57) L3MBTL1LMNAPPARAPPARGLTA4H
SCHEMBL4755605 0.89 L3MBTL1 (0.52) L3MBTL1LMNAPPARAPPARGLTA4H
SCHEMBL2164928 0.87 LTA4H (0.72) PPARAPPARGLTA4HPPARDLAP3
SCHEMBL6732617 0.87 LTA4H (0.72) PPARAPPARGLTA4HPPARDLAP3
SCHEMBL9493387 0.87 L3MBTL1 (0.67) L3MBTL1LMNAPPARAPPARGLTA4H
SCHEMBL5309375 0.87 LTA4H (0.72) PPARAPPARGLTA4HPPARDLAP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 82 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3024816-B1 PPAR-SPARING COMPOUNDS FOR THE TREATMENT OF METABOLIC DISEASES METABOLIC SOLUTIONS DEV CO LLC (US) 2020-06-03 EP disclosed
US-9562012-B2 PPAR-sparing compounds for the treatment of metabolic diseases METABOLIC SOLUTIONS DEVELOPMENT COMPANY, LLC (US) 2017-02-07 US disclosed
US-9562012-B2 PPAR-sparing compounds for the treatment of metabolic diseases METABOLIC SOLUTIONS DEVELOPMENT COMPANY, LLC (US) 2017-02-07 US disclosed
US-20160152570-A1 PPAR-SPARING COMPOUNDS FOR THE TREATMENT OF METABOLIC DISEASES ALZHEIMER'S DRUG DISCOVERY FOUNDATION 2016-06-02 US disclosed
US-20160152570-A1 PPAR-SPARING COMPOUNDS FOR THE TREATMENT OF METABOLIC DISEASES ALZHEIMER'S DRUG DISCOVERY FOUNDATION 2016-06-02 US disclosed
WO-2015013187-A1 PPAR-SPARING COMPOUNDS FOR THE TREATMENT OF METABOLIC DISEASES METABOLIC SOLUTIONS DEVELOPMENT CO., LLC (US) 2015-01-29 WO disclosed
US-7919515-B2 3-phenylpropionic acid derivatives ADAMED SP. Z O.O. (PL) 2011-04-05 US disclosed
US-7919515-B2 3-phenylpropionic acid derivatives ADAMED SP. Z O.O. (PL) 2011-04-05 US disclosed
US-7919515-B2 3-phenylpropionic acid derivatives ADAMED SP. Z O.O. (PL) 2011-04-05 US disclosed
US-7629370-B2 3-phenylpropionic acid derivatives ADAMED SP. Z O.O. (PL) 2009-12-08 US disclosed
CN-1280561-A Amidocarboxylic acid derivatives SANKYO CO (JP) 2001-01-17 CN disclosed
EP-1049684-A1 NOVEL TRICYCLIC COMPOUNDS AND THEIR USE IN MEDICINE; PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-11-08 EP disclosed
WO-2000050414-A1 NOVEL TRICYCLIC COMPOUNDS AND THEIR USE IN MEDICINE; PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITION CONTAINING THEM DR.REDDY'S RESEARCH FOUNDATION (IN) 2000-08-31 WO disclosed
EP-1026149-A1 AMIDOCARBOXYLIC ACID DERIVATIVES Sankyo Company Limited (JP) 2000-08-09 EP disclosed
WO-2000026200-A1 AN IMPROVED PROCESS FOR THE PREPARATION OF NEW ANTIDIABETIC AGENTS DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-05-11 WO disclosed
US-6054453-A HYPOLIPIDEMIC, ANTIHYPERGLYCEMIC USES. REDD'S RESEARCH FOUNDATION (IN) 2000-04-25 US disclosed
WO-1999019313-A1 NOVEL TRICYCLIC COMPOUNDS AND THEIR USE IN MEDICINE; PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 1999-04-22 WO disclosed
US-5391565-A Hypoglycemic agents; antilipemic agents; hypotensive agents BEECHAN GROUP P.L.C. (GB) 1995-02-21 US disclosed
EP-0542816-A1 OXAZOLIDINE DIONE DERIVATIVES BEECHAM GROUP plc (GB) 1993-05-26 EP disclosed
WO-1992002520-A1 OXAZOLIDINE DIONE DERIVATIVES BEECHAM GROUP P.L.C. (GB) 1992-02-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160152570-A1 PPAR-SPARING COMPOUNDS FOR THE TREATMENT OF METABOLIC DISEASES PPARG, PPARA, PPARD L3MBTL1 3403/4885LMNA 2763/4885PPARA 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.