SCHEMBL15979684

SCHEMBL15979684

Cc1ccc(C(=O)CCC(=O)c2cccnc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLOD2 O00469 2/20 0.60
KMT2A Q03164 3/20 0.56
CTNNB1 P35222 1/20 0.56
WNT3A P56704 1/20 0.56
TBXAS1 P24557 1/20 0.54
HDAC1 Q13547 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
NAMPT P43490 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.52
MEN1 O00255 1/20 0.51
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
EGFR P00533 1/20 0.51
PTGS2 P35354 1/20 0.51
ALDH1A1 P00352 2/20 0.51
GAA P10253 2/20 0.50
APP P05067 1/20 0.50
HCAR3 P49019 1/20 0.50
HCAR2 Q8TDS4 1/20 0.50
PLOD3 O60568 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15395342 0.90 PLOD2 (0.75) PLOD2KMT2ATBXAS1HDAC1NAMPT
SCHEMBL7075878 0.88 PLOD2 (0.69) PLOD2KMT2ACTNNB1WNT3ATBXAS1
SCHEMBL9199313 0.86 PLOD2 (0.79) PLOD2KMT2ACTNNB1WNT3ATBXAS1
SCHEMBL1987632 0.83 PLOD2 (0.59) PLOD2KMT2ACTNNB1WNT3ATBXAS1
SCHEMBL15988693 0.83 LMNA (0.70) PLOD2KMT2ATBXAS1NPC1RAB9A
SCHEMBL29861055 0.82 KMT2A (0.55) PLOD2KMT2ANAMPTSMN1; SMN2NPC1
SCHEMBL2511934 0.82 KMT2A (0.55) PLOD2KMT2ANAMPTSMN1; SMN2NPC1
SCHEMBL552724 0.81 PLOD2 (0.61) PLOD2CTNNB1WNT3AHDAC1HDAC8
SCHEMBL29350386 0.81 PLOD2 (0.61) PLOD2CTNNB1WNT3AHDAC1HDAC8
SCHEMBL29450185 0.81 PLOD2 (0.66) PLOD2CTNNB1WNT3ATBXAS1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11673885-B2 γ-diketones as Wnt/β-catenin signaling pathway activators BIOSPLICE THERAPEUTICS, INC. (US) 2023-06-13 US disclosed
US-20180193244-A1 GAMMA-DIKETONES FOR TREATMENT AND PREVENTION OF AGING SKIN AND WRINKLES VICKERS VENTURE FUND VI PTE. LTD. (SG) 2018-07-12 US disclosed
US-9951053-B2 γ-diketones as Wnt/β-catenin signaling pathway activators SAMUMED, LLC (US) 2018-04-24 US disclosed
US-20170260176-A1 GAMMA-DIKETONES AS WNT/BETA -CATENIN SIGNALING PATHWAY ACTIVATORS MED-PATHWAYS II LIMITED (VG) 2017-09-14 US disclosed
US-9533976-B2 γ-diketones as WNT/β-catenin signaling pathway activators SAMUMED, LLC (US) 2017-01-03 US disclosed
US-20160206540-A1 GAMMA-DIKETONES FOR TREATMENT AND PREVENTION OF AGING SKIN AND WRINKLES VICKERS-SPLICE CO-INVESTMENT LLC (KY) 2016-07-21 US disclosed
US-20140243349-A1 GAMMA-DIKETONES AS WNT/BETA -CATENIN SIGNALING PATHWAY ACTIVATORS VICKERS VENTURE FUND VI PTE. LTD. (SG) 2014-08-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180193244-A1 GAMMA-DIKETONES FOR TREATMENT AND PREVENTION OF AGING SKIN AND WRINKLES GLA, DGKG, DGKA PLOD2 178/4885KMT2A 2193/4885CTNNB1 1789/4885
US-20170260176-A1 GAMMA-DIKETONES AS WNT/BETA -CATENIN SIGNALING PATHWAY ACTIVATORS GSK3A, GSK3B, WNT1 PLOD2 1738/4885KMT2A 3457/4885CTNNB1 6/4885
US-20160206540-A1 GAMMA-DIKETONES FOR TREATMENT AND PREVENTION OF AGING SKIN AND WRINKLES GLA, DGKG, DGKA PLOD2 178/4885KMT2A 2193/4885CTNNB1 1789/4885
US-20140243349-A1 GAMMA-DIKETONES AS WNT/BETA -CATENIN SIGNALING PATHWAY ACTIVATORS GSK3A, GSK3B, WNT1 PLOD2 1738/4885KMT2A 3457/4885CTNNB1 6/4885
US-11673885-B2 γ-diketones as Wnt/β-catenin signaling pathway activators GSK3A, GSK3B, WNT1 PLOD2 1746/4885KMT2A 3383/4885CTNNB1 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.