SCHEMBL16004086

SCHEMBL16004086

O=C(c1ccc2c(c1)OCO2)N1CCOc2ccc(COCCc3ccccc3)cc2C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.53
HPGD P15428 6/20 0.53
NPC1 O15118 4/20 0.53
TP53 P04637 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
PKM P14618 2/20 0.48
RAB9A P51151 2/20 0.46
HSD17B10 Q99714 2/20 0.46
TSHR P16473 2/20 0.46
GFER P55789 1/20 0.46
PIK3CA P42336 1/20 0.46
KLF5 Q13887 2/20 0.44
RIPK1 Q13546 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.43
TAS1R3 Q7RTX0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004097 0.87 GPR142 (0.47) PIK3CARIPK1
SCHEMBL16004254 0.86 PIK3CA (0.47) ALDH1A1HPGDNPC1TP53SMN1; SMN2
SCHEMBL16004102 0.83 PIK3CA (0.41) ALDH1A1NPC1RAB9ATSHRPIK3CA
SCHEMBL16004095 0.82 LMNA (0.43) ALDH1A1SMN1; SMN2PIK3CARIPK1LMNA
SCHEMBL16003999 0.82 PIK3CA (0.51) ALDH1A1HPGDNPC1TP53SMN1; SMN2
SCHEMBL16004091 0.78 ALDH1A1 (0.48) ALDH1A1HPGDNPC1SMN1; SMN2RAB9A
SCHEMBL16004297 0.77 FKBP1A (0.51) ALDH1A1HPGDNPC1SMN1; SMN2RAB9A
SCHEMBL16003985 0.76 ATM (0.43) ALDH1A1HPGDTP53PIK3CARIPK1
SCHEMBL16004317 0.76 GPR142 (0.61) ALDH1A1TP53SMN1; SMN2PKMKMT2A
SCHEMBL16004004 0.75 GPR142 (0.49) ALDH1A1HPGDNPC1SMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed